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Alpha2-adrenoreceptors profile modulation. 4. From antagonist to agonist behavior.
J Med Chem. 2008 Jul 24;51(14):4289-99. doi: 10.1021/jm800250z. Epub 2008 Jun 25.
J Med Chem. 2008.
PMID: 18578476
Novel ligands rationally designed for characterizing I2-imidazoline binding sites nature and functions.
Gentili F, Cardinaletti C, Vesprini C, Ghelfi F, Farande A, Giannella M, Piergentili A, Quaglia W, Mattioli L, Perfumi M, Hudson A, Pigini M.
Gentili F, et al. Among authors: farande a.
J Med Chem. 2008 Aug 28;51(16):5130-4. doi: 10.1021/jm800400k. Epub 2008 Jul 29.
J Med Chem. 2008.
PMID: 18661965
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Synthesis and biological evaluation of a novel series of heterobivalent muscarinic ligands based on xanomeline and 1-[3-(4-butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1).
Bonifazi A, Yano H, Del Bello F, Farande A, Quaglia W, Petrelli R, Matucci R, Nesi M, Vistoli G, Ferré S, Piergentili A.
Bonifazi A, et al. Among authors: farande a.
J Med Chem. 2014 Nov 13;57(21):9065-77. doi: 10.1021/jm501173q. Epub 2014 Oct 16.
J Med Chem. 2014.
PMID: 25275964
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Identification of 2-aminopyrimidine derivatives as inhibitors of the canonical Wnt signaling pathway.
Del Bello F, Farande A, Giannella M, Piergentili A, Quaglia W, Benicchi T, Cappelli F, Nencini A, Salerno M, Thomas RJ, Travagli M, Varrone M.
Del Bello F, et al. Among authors: farande a.
Bioorg Med Chem. 2015 Sep 1;23(17):5725-33. doi: 10.1016/j.bmc.2015.07.015. Epub 2015 Jul 17.
Bioorg Med Chem. 2015.
PMID: 26233797
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