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Discovery of novel benzothiophene derivatives as potent and narrow spectrum inhibitors of DYRK1A and DYRK1B.
Bioorg Med Chem Lett. 2022 Jul 15;68:128764. doi: 10.1016/j.bmcl.2022.128764. Epub 2022 May 2.
Bioorg Med Chem Lett. 2022.
PMID: 35504513
Binding and structural analyses of potent inhibitors of the human Ca2+/calmodulin dependent protein kinase kinase 2 (CAMKK2) identified from a collection of commercially-available kinase inhibitors.
Profeta GS, Dos Reis CV, Santiago ADS, Godoi PHC, Fala AM, Wells CI, Sartori R, Salmazo APT, Ramos PZ, Massirer KB, Elkins JM, Drewry DH, Gileadi O, Couñago RM.
Profeta GS, et al. Among authors: fala am.
Sci Rep. 2019 Nov 11;9(1):16452. doi: 10.1038/s41598-019-52795-1.
Sci Rep. 2019.
PMID: 31712618
Free PMC article.
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Development of 2-(4-pyridyl)-benzimidazoles as PKN2 chemical tools to probe cancer.
Scott F, Fala AM, Pennicott LE, Reuillon TD, Massirer KB, Elkins JM, Ward SE.
Scott F, et al. Among authors: fala am.
Bioorg Med Chem Lett. 2020 Apr 15;30(8):127040. doi: 10.1016/j.bmcl.2020.127040. Epub 2020 Feb 17.
Bioorg Med Chem Lett. 2020.
PMID: 32085971
Free PMC article.
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Development of dihydropyrrolopyridinone-based PKN2/PRK2 chemical tools to enable drug discovery.
Scott F, Fala AM, Takarada JE, Ficu MP, Pennicott LE, Reuillon TD, Couñago RM, Massirer KB, Elkins JM, Ward SE.
Scott F, et al. Among authors: fala am.
Bioorg Med Chem Lett. 2022 Mar 15;60:128588. doi: 10.1016/j.bmcl.2022.128588. Epub 2022 Jan 29.
Bioorg Med Chem Lett. 2022.
PMID: 35104640
Free article.
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Identification of inhibitors for the transmembrane Trypanosoma cruzi eIF2α kinase relevant for parasite proliferation.
Marcelino TP, Fala AM, da Silva MM, Souza-Melo N, Malvezzi AM, Klippel AH, Zoltner M, Padilla-Mejia N, Kosto S, Field MC, Burle-Caldas GA, Teixeira SMR, Couñago RM, Massirer KB, Schenkman S.
Marcelino TP, et al. Among authors: fala am.
J Biol Chem. 2023 Jul;299(7):104857. doi: 10.1016/j.jbc.2023.104857. Epub 2023 May 23.
J Biol Chem. 2023.
PMID: 37230387
Free PMC article.
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Human mitochondrial pyruvate carrier 2 as an autonomous membrane transporter.
Nagampalli RSK, Quesñay JEN, Adamoski D, Islam Z, Birch J, Sebinelli HG, Girard RMBM, Ascenção CFR, Fala AM, Pauletti BA, Consonni SR, de Oliveira JF, Silva ACT, Franchini KG, Leme AFP, Silber AM, Ciancaglini P, Moraes I, Dias SMG, Ambrosio ALB.
Nagampalli RSK, et al. Among authors: fala am.
Sci Rep. 2018 Feb 22;8(1):3510. doi: 10.1038/s41598-018-21740-z.
Sci Rep. 2018.
PMID: 29472561
Free PMC article.
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Unsaturated fatty acids as high-affinity ligands of the C-terminal Per-ARNT-Sim domain from the Hypoxia-inducible factor 3α.
Fala AM, Oliveira JF, Adamoski D, Aricetti JA, Dias MM, Dias MVB, Sforça ML, Lopes-de-Oliveira PS, Rocco SA, Caldana C, Dias SMG, Ambrosio ALB.
Fala AM, et al.
Sci Rep. 2015 Aug 3;5:12698. doi: 10.1038/srep12698.
Sci Rep. 2015.
PMID: 26237540
Free PMC article.
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Discovery of pyrazolo[3,4-d]pyrimidines as novel mitogen-activated protein kinase kinase 3 (MKK3) inhibitors.
Takarada JE, Cunha MR, Almeida VM, Vasconcelos SNS, Santiago AS, Godoi PH, Salmazo A, Ramos PZ, Fala AM, de Souza LR, Da Silva IEP, Bengtson MH, Massirer KB, Couñago RM.
Takarada JE, et al. Among authors: fala am.
Bioorg Med Chem. 2024 Jan 15;98:117561. doi: 10.1016/j.bmc.2023.117561. Epub 2023 Dec 20.
Bioorg Med Chem. 2024.
PMID: 38157838
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