Skip to main page content
U.S. flag

An official website of the United States government

Dot gov

The .gov means it’s official.
Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you’re on a federal government site.

Https

The site is secure.
The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.

Access keys NCBI Homepage MyNCBI Homepage Main Content Main Navigation

Search Page

Filters

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

Search Results

238 results

Filters applied: . Clear all
Results are displayed in a computed author sort order. The Results By Year timeline is not available.
Page 1
Design, Synthesis, and Biological Evaluation of 2-Hydroxy-4-phenylthiophene-3-carbonitrile as PD-L1 Antagonist and Its Comparison to Available Small Molecular PD-L1 Inhibitors.
Ważyńska MA, Butera R, Requesens M, Plat A, Zarganes-Tzitzikas T, Neochoritis CG, Plewka J, Skalniak L, Kocik-Krol J, Musielak B, Magiera-Mularz K, Rodriguez I, Blok SN, de Bruyn M, Nijman HW, Elsinga PH, Holak TA, Dömling A. Ważyńska MA, et al. Among authors: elsinga ph. J Med Chem. 2023 Jul 27;66(14):9577-9591. doi: 10.1021/acs.jmedchem.3c00254. Epub 2023 Jul 14. J Med Chem. 2023. PMID: 37450644 Free PMC article.
In vivo responses of human A375M melanoma to a σ ligand: 18F-FDG PET imaging.
Rybczynska AA, de Bruyn M, Ramakrishnan NK, de Jong JR, Elsinga PH, Helfrich W, Dierckx RA, van Waarde A. Rybczynska AA, et al. Among authors: elsinga ph. J Nucl Med. 2013 Sep;54(9):1613-20. doi: 10.2967/jnumed.113.122655. Epub 2013 Aug 12. J Nucl Med. 2013. PMID: 23940303 Free article.
Development of [18F]-labeled pyrazolo[4,3-e]-1,2,4- triazolo[1,5-c]pyrimidine (SCH442416) analogs for the imaging of cerebral adenosine A2A receptors with positron emission tomography.
Khanapur S, Paul S, Shah A, Vatakuti S, Koole MJ, Zijlma R, Dierckx RA, Luurtsema G, Garg P, van Waarde A, Elsinga PH. Khanapur S, et al. Among authors: elsinga ph. J Med Chem. 2014 Aug 14;57(15):6765-80. doi: 10.1021/jm500700y. Epub 2014 Aug 4. J Med Chem. 2014. PMID: 25061687
Synthesis and preclinical evaluation of 2-(2-furanyl)-7-[2-[4-[4-(2-[11C]methoxyethoxy)phenyl]-1-piperazinyl]ethyl]7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine-5-amine ([11C]Preladenant) as a PET tracer for the imaging of cerebral adenosine A2A receptors.
Zhou X, Khanapur S, Huizing AP, Zijlma R, Schepers M, Dierckx RA, van Waarde A, de Vries EF, Elsinga PH. Zhou X, et al. Among authors: elsinga ph. J Med Chem. 2014 Nov 13;57(21):9204-10. doi: 10.1021/jm501065t. Epub 2014 Oct 15. J Med Chem. 2014. PMID: 25279444
MCR Scaffolds Get Hotter with 18F-Labeling.
Zarganes-Tzitzikas T, Clemente GS, Elsinga PH, Dömling A. Zarganes-Tzitzikas T, et al. Among authors: elsinga ph. Molecules. 2019 Apr 4;24(7):1327. doi: 10.3390/molecules24071327. Molecules. 2019. PMID: 30987302 Free PMC article.
Mapping Arginase Expression with 18F-Fluorinated Late-Generation Arginase Inhibitors Derived from Quaternary α-Amino Acids.
Clemente GS, Antunes IF, Kurhade S, van den Berg MPM, Sijbesma JWA, van Waarde A, Buijsman RC, Willemsen-Seegers N, Gosens R, Meurs H, Dömling A, Elsinga PH. Clemente GS, et al. Among authors: elsinga ph. J Nucl Med. 2021 Aug 1;62(8):1163-1170. doi: 10.2967/jnumed.120.255968. Epub 2021 Mar 12. J Nucl Med. 2021. PMID: 33712529 Free article.
Design, Synthesis, and Biological Evaluation of Imidazopyridines as PD-1/PD-L1 Antagonists.
Butera R, Ważyńska M, Magiera-Mularz K, Plewka J, Musielak B, Surmiak E, Sala D, Kitel R, de Bruyn M, Nijman HW, Elsinga PH, Holak TA, Dömling A. Butera R, et al. Among authors: elsinga ph. ACS Med Chem Lett. 2021 Apr 28;12(5):768-773. doi: 10.1021/acsmedchemlett.1c00033. eCollection 2021 May 13. ACS Med Chem Lett. 2021. PMID: 34055224 Free PMC article.
238 results