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New targets for HIV drug discovery.
Puhl AC, Garzino Demo A, Makarov VA, Ekins S. Puhl AC, et al. Among authors: ekins s. Drug Discov Today. 2019 May;24(5):1139-1147. doi: 10.1016/j.drudis.2019.03.013. Epub 2019 Mar 15. Drug Discov Today. 2019. PMID: 30885676 Free PMC article. Review.
Computational mapping tools for drug discovery.
Ivanenkov YA, Savchuk NP, Ekins S, Balakin KV. Ivanenkov YA, et al. Among authors: ekins s. Drug Discov Today. 2009 Aug;14(15-16):767-75. doi: 10.1016/j.drudis.2009.05.016. Epub 2009 Jun 9. Drug Discov Today. 2009. PMID: 19520185 Review.
Alternative business models for drug discovery.
Bunin BA, Ekins S. Bunin BA, et al. Among authors: ekins s. Drug Discov Today. 2011 Aug;16(15-16):643-5. doi: 10.1016/j.drudis.2011.06.012. Epub 2011 Jul 2. Drug Discov Today. 2011. PMID: 21745585 No abstract available.
Mobile apps for chemistry in the world of drug discovery.
Williams AJ, Ekins S, Clark AM, Jack JJ, Apodaca RL. Williams AJ, et al. Among authors: ekins s. Drug Discov Today. 2011 Nov;16(21-22):928-39. doi: 10.1016/j.drudis.2011.09.002. Epub 2011 Sep 6. Drug Discov Today. 2011. PMID: 21924376 Review.
Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG.
Mori G, Chiarelli LR, Esposito M, Makarov V, Bellinzoni M, Hartkoorn RC, Degiacomi G, Boldrin F, Ekins S, de Jesus Lopes Ribeiro AL, Marino LB, Centárová I, Svetlíková Z, Blaško J, Kazakova E, Lepioshkin A, Barilone N, Zanoni G, Porta A, Fondi M, Fani R, Baulard AR, Mikušová K, Alzari PM, Manganelli R, de Carvalho LP, Riccardi G, Cole ST, Pasca MR. Mori G, et al. Among authors: ekins s. Chem Biol. 2015 Jul 23;22(7):917-27. doi: 10.1016/j.chembiol.2015.05.016. Epub 2015 Jun 18. Chem Biol. 2015. PMID: 26097035 Free PMC article.
Learning from the past for TB drug discovery in the future.
Mikušová K, Ekins S. Mikušová K, et al. Among authors: ekins s. Drug Discov Today. 2017 Mar;22(3):534-545. doi: 10.1016/j.drudis.2016.09.025. Epub 2016 Oct 4. Drug Discov Today. 2017. PMID: 27717850 Free PMC article. Review.
371 results