Egerland U - Search Results

1

Fluorine-containing 6,7-dialkoxybiaryl-based inhibitors for phosphodiesterase 10 A: synthesis and in vitro evaluation of inhibitory potency, selectivity, and metabolism.

Schwan G, Barbar Asskar G, Höfgen N, Kubicova L, Funke U, Egerland U, Zahn M, Nieber K, Scheunemann M, Sträter N, Brust P, Briel D. Schwan G, et al. Among authors: egerland u. ChemMedChem. 2014 Jul;9(7):1476-87. doi: 10.1002/cmdc.201300522. Epub 2014 Apr 11. ChemMedChem. 2014. PMID: 24729456

2

Development of highly potent phosphodiesterase 10A (PDE10A) inhibitors: Synthesis and in vitro evaluation of 1,8-dipyridinyl- and 1-pyridinyl-substituted imidazo[1,5-a]quinoxalines.

Wagner S, Scheunemann M, Dipper K, Egerland U, Hoefgen N, Steinbach J, Brust P. Wagner S, et al. Among authors: egerland u. Eur J Med Chem. 2016 Jan 1;107:97-108. doi: 10.1016/j.ejmech.2015.10.028. Epub 2015 Oct 19. Eur J Med Chem. 2016. PMID: 26562545

3

Radiosynthesis and biological evaluation of the new PDE10A radioligand [¹⁸ F]AQ28A.

Wagner S, Teodoro R, Deuther-Conrad W, Kranz M, Scheunemann M, Fischer S, Wenzel B, Egerland U, Hoefgen N, Steinbach J, Brust P. Wagner S, et al. Among authors: egerland u. J Labelled Comp Radiopharm. 2017 Jan;60(1):36-48. doi: 10.1002/jlcr.3471. Epub 2016 Nov 29. J Labelled Comp Radiopharm. 2017. PMID: 27896836

4

Investigation of an ¹⁸F-labelled Imidazopyridotriazine for Molecular Imaging of Cyclic Nucleotide Phosphodiesterase 2A.

Schröder S, Wenzel B, Deuther-Conrad W, Teodoro R, Kranz M, Scheunemann M, Egerland U, Höfgen N, Briel D, Steinbach J, Brust P. Schröder S, et al. Among authors: egerland u. Molecules. 2018 Mar 2;23(3):556. doi: 10.3390/molecules23030556. Molecules. 2018. PMID: 29498659 Free PMC article.

5

Synthesis, 18F-Radiolabelling and Biological Characterization of Novel Fluoroalkylated Triazine Derivatives for in Vivo Imaging of Phosphodiesterase 2A in Brain via Positron Emission Tomography.

Schröder S, Wenzel B, Deuther-Conrad W, Teodoro R, Egerland U, Kranz M, Scheunemann M, Höfgen N, Steinbach J, Brust P. Schröder S, et al. Among authors: egerland u. Molecules. 2015 May 26;20(6):9591-615. doi: 10.3390/molecules20069591. Molecules. 2015. PMID: 26016549 Free PMC article.

6

Synthesis, pharmacology, and structure-activity relationships of novel imidazolones and pyrrolones as modulators of GABAA receptors.

Grunwald C, Rundfeldt C, Lankau HJ, Arnold T, Höfgen N, Dost R, Egerland U, Hofmann HJ, Unverferth K. Grunwald C, et al. Among authors: egerland u. J Med Chem. 2006 Mar 23;49(6):1855-66. doi: 10.1021/jm0509400. J Med Chem. 2006. PMID: 16539371

7

Discovery of imidazo[1,5-a]pyrido[3,2-e]pyrazines as a new class of phosphodiesterase 10A inhibitiors.

Höfgen N, Stange H, Schindler R, Lankau HJ, Grunwald C, Langen B, Egerland U, Tremmel P, Pangalos MN, Marquis KL, Hage T, Harrison BL, Malamas MS, Brandon NJ, Kronbach T. Höfgen N, et al. Among authors: egerland u. J Med Chem. 2010 Jun 10;53(11):4399-411. doi: 10.1021/jm1002793. J Med Chem. 2010. PMID: 20450197

8

[Synthesis of substituted 6-phenylpyrazolo[3,4-d]pyrimidines with potential adenosin-A2A antagonistic activity].

Briel D, Aurich R, Egerland U, Unverferth K. Briel D, et al. Among authors: egerland u. Pharmazie. 2005 Oct;60(10):732-5. Pharmazie. 2005. PMID: 16259118 German.

9

5-(4-Hydroxy-6-methyl-2-oxo-2H-pyran-3-yl)-7-phenyl-2,3,6,7-tetrahydro-1,4-thiazepines as compounds with high affinity at the benzodiazepine binding site on GABA(A) receptors.

Grunwald C, Kronbach C, Egerland U, Schindler R, Dieckmann R, Heinecke K, Höfgen N, Unverferth K. Grunwald C, et al. Among authors: egerland u. Pharmazie. 2011 Feb;66(2):98-104. doi: 10.1002/chin.201125210. Pharmazie. 2011. PMID: 21434570

10

1,5-Disubstituted indazol-3-ols with anti-inflammatory activity.

Schindler R, Fleischhauer I, Höfgen N, Sauer W, Egerland U, Poppe H, Heer S, Szelenyi I, Kutscher B, Engel J. Schindler R, et al. Among authors: egerland u. Arch Pharm (Weinheim). 1998 Jan;331(1):13-21. doi: 10.1002/(SICI)1521-4184(199801)331:1<13::AID-ARDP13>3.0.CO;2-M. Arch Pharm (Weinheim). 1998. PMID: 9507697

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