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An Immunconjugate Vaccine Alters Distribution and Reduces the Antinociceptive, Behavioral and Physiological Effects of Fentanyl in Male and Female Rats.
Pharmaceutics. 2022 Oct 26;14(11):2290. doi: 10.3390/pharmaceutics14112290.
Pharmaceutics. 2022.
PMID: 36365109
Free PMC article.
Fentanyl conjugate vaccine by injected or mucosal delivery with dmLT or LTA1 adjuvants implicates IgA in protection from drug challenge.
Stone AE, Scheuermann SE, Haile CN, Cuny GD, Velasquez ML, Linhuber JP, Duddupudi AL, Vigliaturo JR, Pravetoni M, Kosten TA, Kosten TR, Norton EB.
Stone AE, et al. Among authors: duddupudi al.
NPJ Vaccines. 2021 May 13;6(1):69. doi: 10.1038/s41541-021-00329-0.
NPJ Vaccines. 2021.
PMID: 33986280
Free PMC article.
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Hypervalent Iodine Mediated Oxidative Cyclization of Acrylamide N-Carbamates to 5,5-Disubstituted Oxazolidine-2,4-diones.
Duddupudi AL, Pandey P, Vo H, Welsh CL, Doerksen RJ, Cuny GD.
Duddupudi AL, et al.
J Org Chem. 2020 Jun 5;85(11):7549-7557. doi: 10.1021/acs.joc.0c00581. Epub 2020 May 11.
J Org Chem. 2020.
PMID: 32392063
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Receptor-interacting protein kinase 2 (RIPK2) and nucleotide-binding oligomerization domain (NOD) cell signaling inhibitors based on a 3,5-diphenyl-2-aminopyridine scaffold.
Suebsuwong C, Dai B, Pinkas DM, Duddupudi AL, Li L, Bufton JC, Schlicher L, Gyrd-Hansen M, Hu M, Bullock AN, Degterev A, Cuny GD.
Suebsuwong C, et al. Among authors: duddupudi al.
Eur J Med Chem. 2020 Aug 15;200:112417. doi: 10.1016/j.ejmech.2020.112417. Epub 2020 May 15.
Eur J Med Chem. 2020.
PMID: 32505849
Free PMC article.
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Necroptosis blockade prevents lung injury in severe influenza.
Gautam A, Boyd DF, Nikhar S, Zhang T, Siokas I, Van de Velde LA, Gaevert J, Meliopoulos V, Thapa B, Rodriguez DA, Cai KQ, Yin C, Schnepf D, Beer J, DeAntoneo C, Williams RM, Shubina M, Livingston B, Zhang D, Andrake MD, Lee S, Boda R, Duddupudi AL, Crawford JC, Vogel P, Loch C, Schwemmle M, Fritz LC, Schultz-Cherry S, Green DR, Cuny GD, Thomas PG, Degterev A, Balachandran S.
Gautam A, et al. Among authors: duddupudi al.
Nature. 2024 Apr;628(8009):835-843. doi: 10.1038/s41586-024-07265-8. Epub 2024 Apr 10.
Nature. 2024.
PMID: 38600381
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Pyrimidinyl Biphenylureas: Identification of New Lead Compounds as Allosteric Modulators of the Cannabinoid Receptor CB1.
Khurana L, Fu BQ, Duddupudi AL, Liao YH, Immadi SS, Kendall DA, Lu D.
Khurana L, et al. Among authors: duddupudi al.
J Med Chem. 2017 Feb 9;60(3):1089-1104. doi: 10.1021/acs.jmedchem.6b01448. Epub 2017 Jan 19.
J Med Chem. 2017.
PMID: 28059509
Free PMC article.
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