Dubois LJ - Search Results

1

Experimental Approaches to Identify Selective Picomolar Inhibitors for Carbonic Anhydrase IX.

Kazokaitė-Adomaitienė J, Becker HM, Smirnovienė J, Dubois LJ, Matulis D. Kazokaitė-Adomaitienė J, et al. Among authors: dubois lj. Curr Med Chem. 2021;28(17):3361-3384. doi: 10.2174/0929867327666201102112841. Curr Med Chem. 2021. PMID: 33138744 Review.

2

Imaging the hypoxia surrogate marker CA IX requires expression and catalytic activity for binding fluorescent sulfonamide inhibitors.

Dubois L, Douma K, Supuran CT, Chiu RK, van Zandvoort MA, Pastoreková S, Scozzafava A, Wouters BG, Lambin P. Dubois L, et al. Radiother Oncol. 2007 Jun;83(3):367-73. doi: 10.1016/j.radonc.2007.04.018. Epub 2007 May 14. Radiother Oncol. 2007. PMID: 17502120

3

Hypoxia-induced expression of carbonic anhydrase 9 is dependent on the unfolded protein response.

van den Beucken T, Koritzinsky M, Niessen H, Dubois L, Savelkouls K, Mujcic H, Jutten B, Kopacek J, Pastorekova S, van der Kogel AJ, Lambin P, Voncken W, Rouschop KM, Wouters BG. van den Beucken T, et al. J Biol Chem. 2009 Sep 4;284(36):24204-12. doi: 10.1074/jbc.M109.006510. Epub 2009 Jun 29. J Biol Chem. 2009. PMID: 19564335 Free PMC article.

4

Imaging of CA IX with fluorescent labelled sulfonamides distinguishes hypoxic and (re)-oxygenated cells in a xenograft tumour model.

Dubois L, Lieuwes NG, Maresca A, Thiry A, Supuran CT, Scozzafava A, Wouters BG, Lambin P. Dubois L, et al. Radiother Oncol. 2009 Sep;92(3):423-8. doi: 10.1016/j.radonc.2009.06.019. Epub 2009 Jul 16. Radiother Oncol. 2009. PMID: 19616332

5

Specific inhibition of carbonic anhydrase IX activity enhances the in vivo therapeutic effect of tumor irradiation.

Dubois L, Peeters S, Lieuwes NG, Geusens N, Thiry A, Wigfield S, Carta F, McIntyre A, Scozzafava A, Dogné JM, Supuran CT, Harris AL, Masereel B, Lambin P. Dubois L, et al. Radiother Oncol. 2011 Jun;99(3):424-31. doi: 10.1016/j.radonc.2011.05.045. Epub 2011 Jun 14. Radiother Oncol. 2011. PMID: 21676479 Free article.

6

Targeting carbonic anhydrase IX by nitroimidazole based sulfamides enhances the therapeutic effect of tumor irradiation: a new concept of dual targeting drugs.

Dubois L, Peeters SG, van Kuijk SJ, Yaromina A, Lieuwes NG, Saraya R, Biemans R, Rami M, Parvathaneni NK, Vullo D, Vooijs M, Supuran CT, Winum JY, Lambin P. Dubois L, et al. Radiother Oncol. 2013 Sep;108(3):523-8. doi: 10.1016/j.radonc.2013.06.018. Epub 2013 Jul 9. Radiother Oncol. 2013. PMID: 23849171 Free article.

7

Hypoxia-targeting carbonic anhydrase IX inhibitors by a new series of nitroimidazole-sulfonamides/sulfamides/sulfamates.

Rami M, Dubois L, Parvathaneni NK, Alterio V, van Kuijk SJ, Monti SM, Lambin P, De Simone G, Supuran CT, Winum JY. Rami M, et al. J Med Chem. 2013 Nov 14;56(21):8512-20. doi: 10.1021/jm4009532. Epub 2013 Oct 31. J Med Chem. 2013. PMID: 24128000

8

Development and biological evaluation of ⁹⁹mTc-sulfonamide derivatives for in vivo visualization of CA IX as surrogate tumor hypoxia markers.

Akurathi V, Dubois L, Celen S, Lieuwes NG, Chitneni SK, Cleynhens BJ, Innocenti A, Supuran CT, Verbruggen AM, Lambin P, Bormans GM. Akurathi V, et al. Eur J Med Chem. 2014 Jan;71:374-84. doi: 10.1016/j.ejmech.2013.10.027. Epub 2013 Oct 30. Eur J Med Chem. 2014. PMID: 24378650

9

Evaluation of carbonic anhydrase IX as a therapeutic target for inhibition of breast cancer invasion and metastasis using a series of in vitro breast cancer models.

Ward C, Meehan J, Mullen P, Supuran C, Dixon JM, Thomas JS, Winum JY, Lambin P, Dubois L, Pavathaneni NK, Jarman EJ, Renshaw L, Um IH, Kay C, Harrison DJ, Kunkler IH, Langdon SP. Ward C, et al. Oncotarget. 2015 Sep 22;6(28):24856-70. doi: 10.18632/oncotarget.4498. Oncotarget. 2015. PMID: 26259239 Free PMC article.

10

Synthesis and in Vivo Biological Evaluation of (68)Ga-Labeled Carbonic Anhydrase IX Targeting Small Molecules for Positron Emission Tomography.

Sneddon D, Niemans R, Bauwens M, Yaromina A, van Kuijk SJ, Lieuwes NG, Biemans R, Pooters I, Pellegrini PA, Lengkeek NA, Greguric I, Tonissen KF, Supuran CT, Lambin P, Dubois L, Poulsen SA. Sneddon D, et al. J Med Chem. 2016 Jul 14;59(13):6431-43. doi: 10.1021/acs.jmedchem.6b00623. Epub 2016 Jun 29. J Med Chem. 2016. PMID: 27322137

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

162 results

Search Page