Drag M - Search Results

1

Plasmodium falciparum neutral aminopeptidases: new targets for anti-malarials.

Skinner-Adams TS, Stack CM, Trenholme KR, Brown CL, Grembecka J, Lowther J, Mucha A, Drag M, Kafarski P, McGowan S, Whisstock JC, Gardiner DL, Dalton JP. Skinner-Adams TS, et al. Among authors: drag m. Trends Biochem Sci. 2010 Jan;35(1):53-61. doi: 10.1016/j.tibs.2009.08.004. Epub 2009 Sep 30. Trends Biochem Sci. 2010. PMID: 19796954 Review.

2

X-ray crystal structure and specificity of the Plasmodium falciparum malaria aminopeptidase PfM18AAP.

Sivaraman KK, Oellig CA, Huynh K, Atkinson SC, Poreba M, Perugini MA, Trenholme KR, Gardiner DL, Salvesen G, Drag M, Dalton JP, Whisstock JC, McGowan S. Sivaraman KK, et al. Among authors: drag m. J Mol Biol. 2012 Sep 28;422(4):495-507. doi: 10.1016/j.jmb.2012.06.006. Epub 2012 Jun 16. J Mol Biol. 2012. PMID: 22709581 Free article.

3

Fingerprinting the substrate specificity of M1 and M17 aminopeptidases of human malaria, Plasmodium falciparum.

Poreba M, McGowan S, Skinner-Adams TS, Trenholme KR, Gardiner DL, Whisstock JC, To J, Salvesen GS, Dalton JP, Drag M. Poreba M, et al. Among authors: drag m. PLoS One. 2012;7(2):e31938. doi: 10.1371/journal.pone.0031938. Epub 2012 Feb 16. PLoS One. 2012. PMID: 22359643 Free PMC article.

4

Synthesis and structure-activity relationships of phosphonic arginine mimetics as inhibitors of the M1 and M17 aminopeptidases from Plasmodium falciparum.

Kannan Sivaraman K, Paiardini A, Sieńczyk M, Ruggeri C, Oellig CA, Dalton JP, Scammells PJ, Drag M, McGowan S. Kannan Sivaraman K, et al. Among authors: drag m. J Med Chem. 2013 Jun 27;56(12):5213-7. doi: 10.1021/jm4005972. Epub 2013 Jun 13. J Med Chem. 2013. PMID: 23713488 Free article.

5

Structure and substrate fingerprint of aminopeptidase P from Plasmodium falciparum.

Drinkwater N, Sivaraman KK, Bamert RS, Rut W, Mohamed K, Vinh NB, Scammells PJ, Drag M, McGowan S. Drinkwater N, et al. Among authors: drag m. Biochem J. 2016 Oct 1;473(19):3189-204. doi: 10.1042/BCJ20160550. Epub 2016 Jul 26. Biochem J. 2016. PMID: 27462122

6

Mapping the substrate specificity of the Plasmodium M1 and M17 aminopeptidases.

Malcolm TR, Swiderska KW, Hayes BK, Webb CT, Drag M, Drinkwater N, McGowan S. Malcolm TR, et al. Among authors: drag m. Biochem J. 2021 Jul 16;478(13):2697-2713. doi: 10.1042/BCJ20210172. Biochem J. 2021. PMID: 34133730 Free PMC article.

7

Metallo-aminopeptidase inhibitors.

Mucha A, Drag M, Dalton JP, Kafarski P. Mucha A, et al. Among authors: drag m. Biochimie. 2010 Nov;92(11):1509-29. doi: 10.1016/j.biochi.2010.04.026. Epub 2010 May 10. Biochimie. 2010. PMID: 20457213 Free PMC article. Review.

8

alpha-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases.

Drag M, Grembecka J, Pawełczak M, Kafarski P. Drag M, et al. Eur J Med Chem. 2005 Aug;40(8):764-71. doi: 10.1016/j.ejmech.2005.02.011. Epub 2005 Apr 20. Eur J Med Chem. 2005. PMID: 16122579

9

X-ray crystal structure and specificity of the Toxoplasma gondii ME49 TgAPN2.

Marijanovic EM, Weronika Swiderska K, Andersen J, Aschenbrenner JC, Webb CT, Drag M, Drinkwater N, McGowan S. Marijanovic EM, et al. Among authors: drag m. Biochem J. 2020 Oct 16;477(19):3819-3832. doi: 10.1042/BCJ20200569. Biochem J. 2020. PMID: 32926129 Free PMC article.

10

Chemical target validation studies of aminopeptidase in malaria parasites using alpha-aminoalkylphosphonate and phosphonopeptide inhibitors.

Cunningham E, Drag M, Kafarski P, Bell A. Cunningham E, et al. Among authors: drag m. Antimicrob Agents Chemother. 2008 Sep;52(9):3221-8. doi: 10.1128/AAC.01327-07. Epub 2008 May 5. Antimicrob Agents Chemother. 2008. PMID: 18458130 Free PMC article.

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