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Differential abundance of CK1α provides selectivity for pharmacological CK1α activators to target WNT-dependent tumors.
Sci Signal. 2017 Jun 27;10(485):eaak9916. doi: 10.1126/scisignal.aak9916.
Sci Signal. 2017.
PMID: 28655862
Free PMC article.
A missense mutation in Caenorhabditis elegans prohibitin 2 confers an atypical multidrug resistance.
Zubovych I, Doundoulakis T, Harran PG, Roth MG.
Zubovych I, et al. Among authors: doundoulakis t.
Proc Natl Acad Sci U S A. 2006 Oct 17;103(42):15523-8. doi: 10.1073/pnas.0607338103. Epub 2006 Oct 10.
Proc Natl Acad Sci U S A. 2006.
PMID: 17032754
Free PMC article.
Item in Clipboard
Spirocycloisomerization of tethered alkylidene glycocyamidines: synthesis of a base template common to the palau'amine family of alkaloids.
Garrido-Hernandez H, Nakadai M, Vimolratana M, Li Q, Doundoulakis T, Harran PG.
Garrido-Hernandez H, et al. Among authors: doundoulakis t.
Angew Chem Int Ed Engl. 2005 Jan 21;44(5):765-9. doi: 10.1002/anie.200462069.
Angew Chem Int Ed Engl. 2005.
PMID: 15624220
No abstract available.
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Total Synthesis of (±)-2-Debromohymenin via Gold-Catalyzed Intramolecular Alkyne Hydroarylation.
Singh RP, Bhandari MR, Torres FM, Doundoulakis T, Gout D, Lovely CJ.
Singh RP, et al. Among authors: doundoulakis t.
Org Lett. 2020 May 1;22(9):3412-3417. doi: 10.1021/acs.orglett.0c00883. Epub 2020 Apr 14.
Org Lett. 2020.
PMID: 32286836
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The enantiomeric separation of tetrahydrobenzimidazoles cyclodextrins- and cyclofructans.
Perera S, Na YC, Doundoulakis T, Ngo VJ, Feng Q, Breitbach ZS, Lovely CJ, Armstrong DW.
Perera S, et al. Among authors: doundoulakis t.
Chirality. 2013 Feb;25(2):133-40. doi: 10.1002/chir.22127. Epub 2012 Dec 13.
Chirality. 2013.
PMID: 23238886
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Syntheses of novel myxopyronin B analogs as potential inhibitors of bacterial RNA polymerase.
Lira R, Xiang AX, Doundoulakis T, Biller WT, Agrios KA, Simonsen KB, Webber SE, Sisson W, Aust RM, Shah AM, Showalter RE, Banh VN, Steffy KR, Appleman JR.
Lira R, et al. Among authors: doundoulakis t.
Bioorg Med Chem Lett. 2007 Dec 15;17(24):6797-800. doi: 10.1016/j.bmcl.2007.10.017. Epub 2007 Oct 17.
Bioorg Med Chem Lett. 2007.
PMID: 17980587
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Myxopyronin B analogs as inhibitors of RNA polymerase, synthesis and biological evaluation.
Doundoulakis T, Xiang AX, Lira R, Agrios KA, Webber SE, Sisson W, Aust RM, Shah AM, Showalter RE, Appleman JR, Simonsen KB.
Doundoulakis T, et al.
Bioorg Med Chem Lett. 2004 Nov 15;14(22):5667-72. doi: 10.1016/j.bmcl.2004.08.045.
Bioorg Med Chem Lett. 2004.
PMID: 15482944
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