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Substituted 3-imidazo[1,2-a]pyridin-3-yl- 4-(1,2,3,4-tetrahydro-[1,4]diazepino-[6,7,1-hi]indol-7-yl)pyrrole-2,5-diones as highly selective and potent inhibitors of glycogen synthase kinase-3.
J Med Chem. 2004 Jul 29;47(16):3934-7. doi: 10.1021/jm049768a.
J Med Chem. 2004.
PMID: 15267232
The development of potent and selective bisarylmaleimide GSK3 inhibitors.
Engler TA, Malhotra S, Burkholder TP, Henry JR, Mendel D, Porter WJ, Furness K, Diefenbacher C, Marquart A, Reel JK, Li Y, Clayton J, Cunningham B, McLean J, O'toole JC, Brozinick J, Hawkins E, Misener E, Briere D, Brier RA, Wagner JR, Campbell RM, Anderson BD, Vaughn R, Bennett DB, Meier TI, Cook JA.
Engler TA, et al. Among authors: diefenbacher c.
Bioorg Med Chem Lett. 2005 Feb 15;15(4):899-903. doi: 10.1016/j.bmcl.2004.12.063.
Bioorg Med Chem Lett. 2005.
PMID: 15686883
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Dual angiotensin converting enzyme/thromboxane synthase inhibitors.
Ksander GM, Erion M, Yuan AM, Diefenbacher CG, el-Chehabi L, Cote D, Levens N.
Ksander GM, et al. Among authors: diefenbacher cg.
J Med Chem. 1994 Jun 10;37(12):1823-32. doi: 10.1021/jm00038a011.
J Med Chem. 1994.
PMID: 8021921
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Angiotensin converting enzyme inhibitors: N-substituted D-glutamic acid gamma dipeptides.
Ksander GM, Yuan AM, Diefenbacher CG, Stanton JL.
Ksander GM, et al. Among authors: diefenbacher cg.
J Med Chem. 1985 Nov;28(11):1606-11. doi: 10.1021/jm00149a011.
J Med Chem. 1985.
PMID: 2999395
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Enkephalinase inhibitors. 1. 2,4-Dibenzylglutaric acid derivatives.
Ksander GM, Diefenbacher CG, Yuan AM, Clark F, Sakane Y, Ghai RD.
Ksander GM, et al. Among authors: diefenbacher cg.
J Med Chem. 1989 Dec;32(12):2519-26. doi: 10.1021/jm00132a005.
J Med Chem. 1989.
PMID: 2585440
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Dicarboxylic acid dipeptide neutral endopeptidase inhibitors.
Ksander GM, Ghai RD, deJesus R, Diefenbacher CG, Yuan A, Berry C, Sakane Y, Trapani A.
Ksander GM, et al. Among authors: diefenbacher cg.
J Med Chem. 1995 May 12;38(10):1689-700. doi: 10.1021/jm00010a014.
J Med Chem. 1995.
PMID: 7752193
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Exhaled nitric oxide distinguishes between subgroups of preschool children with respiratory symptoms.
Moeller A, Diefenbacher C, Lehmann A, Rochat M, Brooks-Wildhaber J, Hall GL, Wildhaber JH.
Moeller A, et al. Among authors: diefenbacher c.
J Allergy Clin Immunol. 2008 Mar;121(3):705-9. doi: 10.1016/j.jaci.2007.11.008. Epub 2008 Jan 4.
J Allergy Clin Immunol. 2008.
PMID: 18177695
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