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Design, Synthesis, and Biological Evaluation of a Series of Oxazolone Carboxamides as a Novel Class of Acid Ceramidase Inhibitors.
Caputo S, Di Martino S, Cilibrasi V, Tardia P, Mazzonna M, Russo D, Penna I, Summa M, Bertozzi SM, Realini N, Margaroli N, Migliore M, Ottonello G, Liu M, Lansbury P, Armirotti A, Bertorelli R, Ray SS, Skerlj R, Scarpelli R. Caputo S, et al. Among authors: di martino s. J Med Chem. 2020 Dec 24;63(24):15821-15851. doi: 10.1021/acs.jmedchem.0c01561. Epub 2020 Dec 8. J Med Chem. 2020. PMID: 33290061 Free PMC article.
Synthesis and photocytotoxic activity of [1,2,3]triazolo[4,5-h][1,6]naphthyridines and [1,3]oxazolo[5,4-h][1,6]naphthyridines.
Frasson I, Spanò V, Di Martino S, Nadai M, Doria F, Parrino B, Carbone A, Cascioferro SM, Diana P, Cirrincione G, Freccero M, Barraja P, Richter SN, Montalbano A. Frasson I, et al. Among authors: di martino s. Eur J Med Chem. 2019 Jan 15;162:176-193. doi: 10.1016/j.ejmech.2018.10.071. Epub 2018 Nov 3. Eur J Med Chem. 2019. PMID: 30445266
Second-Generation Non-Covalent NAAA Inhibitors are Protective in a Model of Multiple Sclerosis.
Migliore M Dr, Pontis S Dr, Fuentes de Arriba AL, Realini N, Torrente E, Armirotti A, Romeo E, Di Martino S, Russo D, Pizzirani D, Summa M, Lanfranco M, Ottonello G, Busquet P, Jung KM, Garcia-Guzman M, Heim R, Scarpelli R, Piomelli D. Migliore M Dr, et al. Among authors: di martino s. Angew Chem Int Ed Engl. 2016 Sep 5;55(37):11193-11197. doi: 10.1002/anie.201603746. Epub 2016 Jul 12. Angew Chem Int Ed Engl. 2016. PMID: 27404798 Free PMC article.
Lead Optimization of Benzoxazolone Carboxamides as Orally Bioavailable and CNS Penetrant Acid Ceramidase Inhibitors.
Di Martino S, Tardia P, Cilibrasi V, Caputo S, Mazzonna M, Russo D, Penna I, Realini N, Margaroli N, Migliore M, Pizzirani D, Ottonello G, Bertozzi SM, Armirotti A, Nguyen D, Sun Y, Bongarzone ER, Lansbury P, Liu M, Skerlj R, Scarpelli R. Di Martino S, et al. J Med Chem. 2020 Apr 9;63(7):3634-3664. doi: 10.1021/acs.jmedchem.9b02004. Epub 2020 Mar 26. J Med Chem. 2020. PMID: 32176488 Free PMC article.
Thymosin beta4 targeting impairs tumorigenic activity of colon cancer stem cells.
Ricci-Vitiani L, Mollinari C, di Martino S, Biffoni M, Pilozzi E, Pagliuca A, de Stefano MC, Circo R, Merlo D, De Maria R, Garaci E. Ricci-Vitiani L, et al. Among authors: di martino s. FASEB J. 2010 Nov;24(11):4291-301. doi: 10.1096/fj.10-159970. Epub 2010 Jun 21. FASEB J. 2010. PMID: 20566622
Therapeutic implications of colon cancer stem cells.
Fabrizi E, di Martino S, Pelacchi F, Ricci-Vitiani L. Fabrizi E, et al. Among authors: di martino s. World J Gastroenterol. 2010 Aug 21;16(31):3871-7. doi: 10.3748/wjg.v16.i31.3871. World J Gastroenterol. 2010. PMID: 20712047 Free PMC article. Review.
The transient receptor potential vanilloid-2 cation channel impairs glioblastoma stem-like cell proliferation and promotes differentiation.
Morelli MB, Nabissi M, Amantini C, Farfariello V, Ricci-Vitiani L, di Martino S, Pallini R, Larocca LM, Caprodossi S, Santoni M, De Maria R, Santoni G. Morelli MB, et al. Among authors: di martino s. Int J Cancer. 2012 Oct 1;131(7):E1067-77. doi: 10.1002/ijc.27588. Epub 2012 Apr 27. Int J Cancer. 2012. PMID: 22492283 Free article.
137 results