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Metformin Impedes Oxidation of LDL In Vitro.
Pharmaceutics. 2023 Aug 9;15(8):2111. doi: 10.3390/pharmaceutics15082111.
Pharmaceutics. 2023.
PMID: 37631325
Free PMC article.
Macrocyclization as a Source of Desired Polypharmacology. Discovery of Triple PI3K/mTOR/PIM Inhibitors.
Martínez-González S, Alvarez RM, Martín JI, García AB, Riesco-Fagundo C, Varela C, Rodríguez Hergueta A, González Cantalapiedra E, Albarrán MI, Gómez-Casero E, Cebriá A, Aguirre E, Ajenjo N, Cebrián D, Di Geronimo B, Cunningham D, O'Neill M, Dave HPG, Blanco-Aparicio C, Pastor J.
Martínez-González S, et al. Among authors: di geronimo b.
ACS Med Chem Lett. 2021 Nov 2;12(11):1794-1801. doi: 10.1021/acsmedchemlett.1c00412. eCollection 2021 Nov 11.
ACS Med Chem Lett. 2021.
PMID: 34795869
Free PMC article.
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Corrigendum to <' Omipalisib inspired macrocycles as dual PI3K/mTOR inhibitors' [Eur. J. Med. Chem. 211 (2021), 113109].
Alvarez RM, García AB, Riesco-Fagundo C, Martín JI, Varela C, Rodríguez Hergueta A, González Cantalapiedra E, Oyarzabal J, Di Geronimo B, Lorenzo M, Albarrán MI, Cebriá A, Cebrián D, Martínez-González S, Blanco-Aparicio C, Pastor J.
Alvarez RM, et al. Among authors: di geronimo b.
Eur J Med Chem. 2021 Nov 15;224:113703. doi: 10.1016/j.ejmech.2021.113703. Epub 2021 Jul 17.
Eur J Med Chem. 2021.
PMID: 34284231
No abstract available.
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Omipalisib inspired macrocycles as dual PI3K/mTOR inhibitors.
Álvarez RM, García AB, Riesco-Fagundo C, Martín JI, Varela C, Rodríguez Hergueta A, González Cantalapiedra E, Oyarzabal J, Di Geronimo B, Lorenzo M, Albarrán MI, Cebriá A, Cebrián D, Martínez-González S, Blanco-Aparicio C, Pastor J.
Álvarez RM, et al. Among authors: di geronimo b.
Eur J Med Chem. 2021 Feb 5;211:113109. doi: 10.1016/j.ejmech.2020.113109. Epub 2020 Dec 18.
Eur J Med Chem. 2021.
PMID: 33360802
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Pyrrolo[1,2-a]quinoxalines: Insulin Mimetics that Exhibit Potent and Selective Inhibition against Protein Tyrosine Phosphatase 1B.
García-Marín J, Griera M, Sánchez-Alonso P, Di Geronimo B, Mendicuti F, Rodríguez-Puyol M, Alajarín R, de Pascual-Teresa B, Vaquero JJ, Rodríguez-Puyol D.
García-Marín J, et al. Among authors: di geronimo b.
ChemMedChem. 2020 Oct 5;15(19):1788-1801. doi: 10.1002/cmdc.202000446. Epub 2020 Sep 10.
ChemMedChem. 2020.
PMID: 32909701
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Disulfide Engineered Lipase to Enhance the Catalytic Activity: A Structure-Based Approach on BTL2.
Godoy CA, Klett J, Di Geronimo B, Hermoso JA, Guisán JM, Carrasco-López C.
Godoy CA, et al. Among authors: di geronimo b.
Int J Mol Sci. 2019 Oct 23;20(21):5245. doi: 10.3390/ijms20215245.
Int J Mol Sci. 2019.
PMID: 31652673
Free PMC article.
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Pharmacological inhibition of Receptor Protein Tyrosine Phosphatase β/ζ (PTPRZ1) modulates behavioral responses to ethanol.
Fernández-Calle R, Vicente-Rodríguez M, Pastor M, Gramage E, Di Geronimo B, Zapico JM, Coderch C, Pérez-García C, Lasek AW, de Pascual-Teresa B, Ramos A, Herradón G.
Fernández-Calle R, et al. Among authors: di geronimo b.
Neuropharmacology. 2018 Jul 15;137:86-95. doi: 10.1016/j.neuropharm.2018.04.027. Epub 2018 May 9.
Neuropharmacology. 2018.
PMID: 29753117
Free PMC article.
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Development of inhibitors of receptor protein tyrosine phosphatase β/ζ (PTPRZ1) as candidates for CNS disorders.
Pastor M, Fernández-Calle R, Di Geronimo B, Vicente-Rodríguez M, Zapico JM, Gramage E, Coderch C, Pérez-García C, Lasek AW, Puchades-Carrasco L, Pineda-Lucena A, de Pascual-Teresa B, Herradón G, Ramos A.
Pastor M, et al. Among authors: di geronimo b.
Eur J Med Chem. 2018 Jan 20;144:318-329. doi: 10.1016/j.ejmech.2017.11.080. Epub 2017 Nov 28.
Eur J Med Chem. 2018.
PMID: 29275231
Free PMC article.
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