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Synthetic heterocyclic candidates as promising α-glucosidase inhibitors: An overview.
Eur J Med Chem. 2019 Aug 15;176:343-377. doi: 10.1016/j.ejmech.2019.04.025. Epub 2019 Apr 30.
Eur J Med Chem. 2019.
PMID: 31112894
Review.
Flavone-1,2,3-triazole derivatives as potential α-glucosidase inhibitors: Synthesis, enzyme inhibition, kinetic analysis and molecular docking study.
Dhameja M, Kumar H, Kurella S, Uma A, Gupta P.
Dhameja M, et al.
Bioorg Chem. 2022 Oct;127:106028. doi: 10.1016/j.bioorg.2022.106028. Epub 2022 Jul 16.
Bioorg Chem. 2022.
PMID: 35868105
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Synthesis of 1,2,3-triazole-1,3,4-thiadiazole hybrids as novel α-glucosidase inhibitors by in situ azidation/click assembly.
Kumar H, Dhameja M, Kurella S, Uma A, Gupta P.
Kumar H, et al. Among authors: dhameja m.
Arch Pharm (Weinheim). 2023 Aug;356(8):e2300145. doi: 10.1002/ardp.202300145. Epub 2023 May 26.
Arch Pharm (Weinheim). 2023.
PMID: 37236165
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Acute Administration of Ojeok-san Ameliorates Pain-like Behaviors in Pre-Clinical Models of Inflammatory Bowel Diseases.
Patton EA, Cunningham P, Noneman M, Helms HP, Martinez-Muniz G, Sumal AS, Dhameja MK, Unger CA, Alahdami AK, Enos RT, Chatzistamou I, Velázquez KT.
Patton EA, et al. Among authors: dhameja mk.
Nutrients. 2023 Mar 23;15(7):1559. doi: 10.3390/nu15071559.
Nutrients. 2023.
PMID: 37049400
Free PMC article.
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Inhibition of α-glucosidase enzyme by 'click'-inspired pharmacophore framework 1,3,4-thiadiazole-1,2,3-triazole hybrids.
Dhameja M, Kumar H, Kurella S, Singh R, Uma A, Gupta P.
Dhameja M, et al.
Future Med Chem. 2023 Feb;15(4):345-363. doi: 10.4155/fmc-2022-0289. Epub 2023 Mar 21.
Future Med Chem. 2023.
PMID: 36942781
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