Debevec G - Search Results

1

Identification of Bis-Cyclic Guanidines as Antiplasmodial Compounds from Positional Scanning Mixture-Based Libraries.

Perry DL Jr, Roberts BF, Debevec G, Michaels HA, Chakrabarti D, Nefzi A. Perry DL Jr, et al. Among authors: debevec g. Molecules. 2019 Mar 20;24(6):1100. doi: 10.3390/molecules24061100. Molecules. 2019. PMID: 30897744 Free PMC article.

2

Scaffold Ranking and Positional Scanning Identify Novel Neurite Outgrowth Promoters with Nanomolar Potency.

Al-Ali H, Debevec G, Santos RG, Houghten RA, Davis JC, Nefzi A, Lemmon VP, Bixby JL, Giulianotti MA. Al-Ali H, et al. Among authors: debevec g. ACS Med Chem Lett. 2018 Sep 24;9(10):1057-1062. doi: 10.1021/acsmedchemlett.8b00425. eCollection 2018 Oct 11. ACS Med Chem Lett. 2018. PMID: 30344917 Free PMC article.

3

A novel method for the determination of isokinetic ratios and its application in the synthesis of two new positional scanning libraries.

Giulianotti MA, Debevec G, Santos RG, Maida LE, Chen W, Ou L, Yu Y, Dooley CT, Houghten RA. Giulianotti MA, et al. Among authors: debevec g. ACS Comb Sci. 2012 Sep 10;14(9):503-12. doi: 10.1021/co300060s. Epub 2012 Aug 28. ACS Comb Sci. 2012. PMID: 22913403 Free PMC article.

4

Fluorescent mu selective opioid ligands from a mixture based cyclic peptide library.

Li Y, Dooley CT, Misler JA, Debevec G, Giulianotti MA, Cazares ME, Maida L, Houghten RA. Li Y, et al. Among authors: debevec g. ACS Comb Sci. 2012 Dec 10;14(12):673-9. doi: 10.1021/co300110t. Epub 2012 Nov 8. ACS Comb Sci. 2012. PMID: 23110623 Free PMC article.

5

Identification of a small molecule inhibitor of the aminoglycoside 6'-N-acetyltransferase type Ib [AAC(6')-Ib] using mixture-based combinatorial libraries.

Tran T, Chiem K, Jani S, Arivett BA, Lin DL, Lad R, Jimenez V, Farone MB, Debevec G, Santos R, Giulianotti M, Pinilla C, Tolmasky ME. Tran T, et al. Among authors: debevec g. Int J Antimicrob Agents. 2018 May;51(5):752-761. doi: 10.1016/j.ijantimicag.2018.01.019. Epub 2018 Feb 2. Int J Antimicrob Agents. 2018. PMID: 29410367 Free PMC article.

6

Identification of small molecules by screening a mixture-based scaffold compound library for treatment of alpha-1 antitrypsin deficiency.

Zhang X, Santos R, Debevec G, Li D, Schutte R, Pham K, Liu C, Ostrov DA, Giulianotti M. Zhang X, et al. Among authors: debevec g. Biochem Biophys Res Commun. 2020 Jun 18;527(1):317-323. doi: 10.1016/j.bbrc.2020.04.037. Epub 2020 May 11. Biochem Biophys Res Commun. 2020. PMID: 32446387

7

Libraries from Libraries: A Series of Sulfonamide Linked Heterocycles Derived from the Same Scaffold.

Debevec G, Chen W, Yu Y, Houghten RA, Giulianotti MA. Debevec G, et al. Tetrahedron Lett. 2013 Aug 7;54(32):10.1016/j.tetlet.2013.06.003. doi: 10.1016/j.tetlet.2013.06.003. Tetrahedron Lett. 2013. PMID: 24363466 Free PMC article.

8

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput "Unbiased" Screening Campaign.

Doering SR, Freeman K, Debevec G, Geer P, Santos RG, Lavoi TM, Giulianotti MA, Pinilla C, Appel JR, Houghten RA, Ericson MD, Haskell-Luevano C. Doering SR, et al. Among authors: debevec g. J Med Chem. 2021 May 13;64(9):5577-5592. doi: 10.1021/acs.jmedchem.0c02041. Epub 2021 Apr 22. J Med Chem. 2021. PMID: 33886285 Free PMC article.

9

Highly Selective and Potent α4β2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats.

Wu J, Cippitelli A, Zhang Y, Debevec G, Schoch J, Ozawa A, Yu Y, Liu H, Chen W, Houghten RA, Welmaker GS, Giulianotti MA, Toll L. Wu J, et al. Among authors: debevec g. J Med Chem. 2017 Dec 28;60(24):10092-10104. doi: 10.1021/acs.jmedchem.7b01250. Epub 2017 Dec 13. J Med Chem. 2017. PMID: 29178785 Free PMC article.

10

A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation.

Sammons RM, Perry NA, Li Y, Cho EJ, Piserchio A, Zamora-Olivares DP, Ghose R, Kaoud TS, Debevec G, Bartholomeusz C, Gurevich VV, Iverson TM, Giulianotti M, Houghten RA, Dalby KN. Sammons RM, et al. Among authors: debevec g. ACS Chem Biol. 2019 Jun 21;14(6):1183-1194. doi: 10.1021/acschembio.9b00093. Epub 2019 May 13. ACS Chem Biol. 2019. PMID: 31058487 Free PMC article.

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