Halogenation of a capsaicin analogue leads to novel vanilloid TRPV1 receptor antagonists.
Appendino G, Harrison S, De Petrocellis L, Daddario N, Bianchi F, Schiano Moriello A, Trevisani M, Benvenuti F, Geppetti P, Di Marzo V.
Appendino G, et al. Among authors: de petrocellis l.
Br J Pharmacol. 2003 Aug;139(8):1417-24. doi: 10.1038/sj.bjp.0705387.
Br J Pharmacol. 2003.
PMID: 12922928
Free PMC article.