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Page 1
Preliminary in vitro evaluation of the anti-proliferative activity of guanylhydrazone derivatives.
França PH, Da Silva-Júnior EF, Aquino PG, Santana AE, Ferro JN, De Oliveira Barreto E, Do Ó Pessoa C, Meira AS, De Aquino TM, Alexandre-Moreira MS, Schmitt M, De Araújo-Júnior JX. França PH, et al. Among authors: de araujo junior jx, de oliveira barreto e, de aquino tm, aquino pg. Acta Pharm. 2016 Mar;66(1):129-37. doi: 10.1515/acph-2016-0015. Acta Pharm. 2016. PMID: 26959549 Free article.
The influence of N-alkyl chains in benzoyl-thiourea derivatives on urease inhibition: Soil studies and biophysical and theoretical investigations on the mechanism of interaction.
Tavares MC, Dos Santos Nascimento IJ, de Aquino TM, de Oliveira Brito T, Macedo F Jr, Modolo LV, de Fátima Â, Santos JCC. Tavares MC, et al. Among authors: de aquino tm. Biophys Chem. 2023 Aug;299:107042. doi: 10.1016/j.bpc.2023.107042. Epub 2023 May 24. Biophys Chem. 2023. PMID: 37263179
Dynamic Simulation, Docking and DFT Studies Applied to a Set of Anti-Acetylcholinesterase Inhibitors in the enzyme β-Secretase (BACE-1): An Important Therapeutic Target in Alzheimer`s disease.
Silva-Junior EF, Barcellos Franca PH, Quintans-Junior LJ, Mendonca-Junior FJB, Scotti L, Scotti MT, de Aquino TM, de Araujo-Junior JX. Silva-Junior EF, et al. Among authors: de araujo junior jx, de aquino tm. Curr Comput Aided Drug Des. 2017 Nov 10;13(4):266-274. doi: 10.2174/1573409913666170406150905. Curr Comput Aided Drug Des. 2017. PMID: 28382866
Molecular Docking Studies Applied to a Dataset of Cruzain Inhibitors.
da Silva-Junior EF, Barcellos Franca PH, Ribeiro FF, Bezerra Mendonca-Junior FJ, Scotti L, Scotti MT, de Aquino TM, de Araujo-Junior JX. da Silva-Junior EF, et al. Among authors: de araujo junior jx, de aquino tm. Curr Comput Aided Drug Des. 2018;14(1):68-78. doi: 10.2174/1573409913666170519112758. Curr Comput Aided Drug Des. 2018. PMID: 28523999
Aminoguanidine hydrazones (AGH's) as modulators of norfloxacin resistance in Staphylococcus aureus that overexpress NorA efflux pump.
Dantas N, de Aquino TM, de Araújo-Júnior JX, da Silva-Júnior E, Gomes EA, Gomes AAS, Siqueira-Júnior JP, Mendonça Junior FJB. Dantas N, et al. Among authors: de araujo junior jx, de aquino tm. Chem Biol Interact. 2018 Jan 25;280:8-14. doi: 10.1016/j.cbi.2017.12.009. Epub 2017 Dec 5. Chem Biol Interact. 2018. PMID: 29208359
Synthesis and evaluation of the antibiotic and adjuvant antibiotic potential of organotin(IV) derivatives.
Barbosa ASL, Guedes JS, da Silva DR, Meneghetti SMP, Meneghetti MR, da Silva AE, de Araujo MV, Alexandre-Moreira MS, de Aquino TM, de Siqueira Junior JP, de Araújo RSA, da Cruz RMD, Mendonça-Junior FJB. Barbosa ASL, et al. Among authors: de aquino tm, de siqueira junior jp, de araujo rsa, de araujo mv. J Inorg Biochem. 2018 Mar;180:80-88. doi: 10.1016/j.jinorgbio.2017.12.004. Epub 2017 Dec 8. J Inorg Biochem. 2018. PMID: 29247870
Annonalide and derivatives: Semisynthesis, cytotoxic activities and studies on interaction of annonalide with DNA.
Marques RA, Gomes AOCV, de Brito MV, Dos Santos ALP, da Silva GS, de Lima LB, Nunes FM, de Mattos MC, de Oliveira FCE, do Ó Pessoa C, de Moraes MO, de Fátima Â, Franco LL, Silva MM, Dantas MDA, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, de Oliveira MCF, Leslie Gunatilaka AA. Marques RA, et al. Among authors: de araujo junior jx, de aquino tm, de oliveira mcf, de lima lb, de mattos mc, de moraes mo, de fatima a, de oliveira fce, de brito mv. J Photochem Photobiol B. 2018 Feb;179:156-166. doi: 10.1016/j.jphotobiol.2018.01.016. Epub 2018 Feb 3. J Photochem Photobiol B. 2018. PMID: 29413989
Evidence for the involvement of TNF-α, IL-1β and IL-10 in the antinociceptive and anti-inflammatory effects of indole-3-guanylhydrazone hydrochloride, an aromatic aminoguanidine, in rodents.
Sandes SMS, Heimfarth L, Brito RG, Santos PL, Gouveia DN, Carvalho AMS, Quintans JSS, da Silva-Júnior EF, de Aquino TM, França PHB, de Araújo-Júnior JX, Albuquerque-Júnior RLC, Zengin G, Schmitt M, Bourguignon JJ, Quintans-Júnior LJ. Sandes SMS, et al. Among authors: de araujo junior jx, de aquino tm. Chem Biol Interact. 2018 Apr 25;286:1-10. doi: 10.1016/j.cbi.2018.02.026. Epub 2018 Feb 27. Chem Biol Interact. 2018. PMID: 29499192
Highly functionalized piperidines: Free radical scavenging, anticancer activity, DNA interaction and correlation with biological activity.
Das S, da Silva CJ, Silva MM, Dantas MDA, de Fátima Â, Góis Ruiz ALT, da Silva CM, de Carvalho JE, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, Brahmachari G, Modolo LV. Das S, et al. Among authors: de araujo junior jx, de aquino tm, de fatima a, de carvalho je. J Adv Res. 2017 Oct 31;9:51-61. doi: 10.1016/j.jare.2017.10.010. eCollection 2018 Jan. J Adv Res. 2017. PMID: 30046486 Free PMC article.
Correlation between DNA/HSA-interactions and antimalarial activity of acridine derivatives: Proposing a possible mechanism of action.
de M Silva M, Macedo TS, Teixeira HMP, Moreira DRM, Soares MBP, da C Pereira AL, de L Serafim V, Mendonça-Júnior FJB, do Carmo A de Lima M, de Moura RO, da Silva-Júnior EF, de Araújo-Júnior JX, de A Dantas MD, de O O Nascimento E, Maciel TMS, de Aquino TM, Figueiredo IM, Santos JCC. de M Silva M, et al. Among authors: de araujo junior jx, de o o nascimento e, de moura ro, de aquino tm, de a dantas md, de l serafim v. J Photochem Photobiol B. 2018 Dec;189:165-175. doi: 10.1016/j.jphotobiol.2018.10.016. Epub 2018 Oct 19. J Photochem Photobiol B. 2018. PMID: 30366283
41 results