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Engineered anti-inflammatory peptides inspired by mapping an evasin-chemokine interaction.
J Biol Chem. 2020 Aug 7;295(32):10926-10939. doi: 10.1074/jbc.RA120.014103. Epub 2020 May 29.
J Biol Chem. 2020.
PMID: 32471866
Free PMC article.
Structures of mammalian ER α-glucosidase II capture the binding modes of broad-spectrum iminosugar antivirals.
Caputo AT, Alonzi DS, Marti L, Reca IB, Kiappes JL, Struwe WB, Cross A, Basu S, Lowe ED, Darlot B, Santino A, Roversi P, Zitzmann N.
Caputo AT, et al. Among authors: darlot b.
Proc Natl Acad Sci U S A. 2016 Aug 9;113(32):E4630-8. doi: 10.1073/pnas.1604463113. Epub 2016 Jul 26.
Proc Natl Acad Sci U S A. 2016.
PMID: 27462106
Free PMC article.
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Structural Insights into the Broad-Spectrum Antiviral Target Endoplasmic Reticulum Alpha-Glucosidase II.
Caputo AT, Alonzi DS, Kiappes JL, Struwe WB, Cross A, Basu S, Darlot B, Roversi P, Zitzmann N.
Caputo AT, et al. Among authors: darlot b.
Adv Exp Med Biol. 2018;1062:265-276. doi: 10.1007/978-981-10-8727-1_19.
Adv Exp Med Biol. 2018.
PMID: 29845539
Review.
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Fragment expansion with NUDELs - poised DNA-encoded libraries.
Salvini CLA, Darlot B, Davison J, Martin MP, Tudhope SJ, Turberville S, Kawamura A, Noble MEM, Wedge SR, Crawford JJ, Waring MJ.
Salvini CLA, et al. Among authors: darlot b.
Chem Sci. 2023 Jul 12;14(31):8288-8294. doi: 10.1039/d3sc01171b. eCollection 2023 Aug 9.
Chem Sci. 2023.
PMID: 37564419
Free PMC article.
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Crystal polymorphism in fragment-based lead discovery of ligands of the catalytic domain of UGGT, the glycoprotein folding quality control checkpoint.
Caputo AT, Ibba R, Le Cornu JD, Darlot B, Hensen M, Lipp CB, Marcianò G, Vasiljević S, Zitzmann N, Roversi P.
Caputo AT, et al. Among authors: darlot b.
Front Mol Biosci. 2022 Dec 14;9:960248. doi: 10.3389/fmolb.2022.960248. eCollection 2022.
Front Mol Biosci. 2022.
PMID: 36589243
Free PMC article.
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