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Page 1
Molecular Docking Studies Applied to a Dataset of Cruzain Inhibitors.
da Silva-Junior EF, Barcellos Franca PH, Ribeiro FF, Bezerra Mendonca-Junior FJ, Scotti L, Scotti MT, de Aquino TM, de Araujo-Junior JX. da Silva-Junior EF, et al. Curr Comput Aided Drug Des. 2018;14(1):68-78. doi: 10.2174/1573409913666170519112758. Curr Comput Aided Drug Des. 2018. PMID: 28523999
Annonalide and derivatives: Semisynthesis, cytotoxic activities and studies on interaction of annonalide with DNA.
Marques RA, Gomes AOCV, de Brito MV, Dos Santos ALP, da Silva GS, de Lima LB, Nunes FM, de Mattos MC, de Oliveira FCE, do Ó Pessoa C, de Moraes MO, de Fátima Â, Franco LL, Silva MM, Dantas MDA, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, de Oliveira MCF, Leslie Gunatilaka AA. Marques RA, et al. J Photochem Photobiol B. 2018 Feb;179:156-166. doi: 10.1016/j.jphotobiol.2018.01.016. Epub 2018 Feb 3. J Photochem Photobiol B. 2018. PMID: 29413989
Evidence for the involvement of TNF-α, IL-1β and IL-10 in the antinociceptive and anti-inflammatory effects of indole-3-guanylhydrazone hydrochloride, an aromatic aminoguanidine, in rodents.
Sandes SMS, Heimfarth L, Brito RG, Santos PL, Gouveia DN, Carvalho AMS, Quintans JSS, da Silva-Júnior EF, de Aquino TM, França PHB, de Araújo-Júnior JX, Albuquerque-Júnior RLC, Zengin G, Schmitt M, Bourguignon JJ, Quintans-Júnior LJ. Sandes SMS, et al. Chem Biol Interact. 2018 Apr 25;286:1-10. doi: 10.1016/j.cbi.2018.02.026. Epub 2018 Feb 27. Chem Biol Interact. 2018. PMID: 29499192
Highly functionalized piperidines: Free radical scavenging, anticancer activity, DNA interaction and correlation with biological activity.
Das S, da Silva CJ, Silva MM, Dantas MDA, de Fátima Â, Góis Ruiz ALT, da Silva CM, de Carvalho JE, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, Brahmachari G, Modolo LV. Das S, et al. J Adv Res. 2017 Oct 31;9:51-61. doi: 10.1016/j.jare.2017.10.010. eCollection 2018 Jan. J Adv Res. 2017. PMID: 30046486 Free PMC article.
Correlation between DNA/HSA-interactions and antimalarial activity of acridine derivatives: Proposing a possible mechanism of action.
de M Silva M, Macedo TS, Teixeira HMP, Moreira DRM, Soares MBP, da C Pereira AL, de L Serafim V, Mendonça-Júnior FJB, do Carmo A de Lima M, de Moura RO, da Silva-Júnior EF, de Araújo-Júnior JX, de A Dantas MD, de O O Nascimento E, Maciel TMS, de Aquino TM, Figueiredo IM, Santos JCC. de M Silva M, et al. J Photochem Photobiol B. 2018 Dec;189:165-175. doi: 10.1016/j.jphotobiol.2018.10.016. Epub 2018 Oct 19. J Photochem Photobiol B. 2018. PMID: 30366283
5-Nitro-Thiophene-Thiosemicarbazone Derivatives Present Antitumor Activity Mediated by Apoptosis and DNA Intercalation.
Roque Marques KM, do Desterro MR, de Arruda SM, de Araújo Neto LN, do Carmo Alves de Lima M, de Almeida SMV, da Silva ECD, de Aquino TM, da Silva-Júnior EF, de Araújo-Júnior JX, de M Silva M, de A Dantas MD, Santos JCC, Figueiredo IM, Bazin MA, Marchand P, da Silva TG, Mendonça Junior FJB. Roque Marques KM, et al. Curr Top Med Chem. 2019;19(13):1075-1091. doi: 10.2174/1568026619666190621120304. Curr Top Med Chem. 2019. PMID: 31223089
Indole-3-guanylhydrazone hydrochloride mitigates long-term cognitive impairment in a neonatal sepsis model with involvement of MAPK and NFκB pathways.
Heimfarth L, Carvalho AMS, Quintans JSS, Pereira EWM, Lima NT, Bezerra Carvalho MT, Barreto RSS, Moreira JCF, da Silva-Júnior EF, Schmitt M, Bourguignon JJ, de Aquino TM, Araújo-Júnior JX, Quintans-Júnior LJ. Heimfarth L, et al. Neurochem Int. 2020 Mar;134:104647. doi: 10.1016/j.neuint.2019.104647. Epub 2019 Dec 23. Neurochem Int. 2020. PMID: 31877349
51 results