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7 results
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New m-calpain substrate-based azapeptide inhibitors.
J Pept Sci. 2013 Jun;19(6):370-6. doi: 10.1002/psc.2511. Epub 2013 Apr 24.
J Pept Sci. 2013.
PMID: 23613308
Modulators of calpain activity: inhibitors and activators as potential drugs.
Dókus LE, Yousef M, Bánóczi Z.
Dókus LE, et al.
Expert Opin Drug Discov. 2020 Apr;15(4):471-486. doi: 10.1080/17460441.2020.1722638. Epub 2020 Feb 5.
Expert Opin Drug Discov. 2020.
PMID: 32022614
Review.
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Probing of primed and unprimed sites of calpains: Design, synthesis and evaluation of epoxysuccinyl-peptide derivatives as selective inhibitors.
Dókus LE, Menyhárd DK, Tantos Á, Hudecz F, Bánóczi Z.
Dókus LE, et al.
Eur J Med Chem. 2014 Jul 23;82:274-80. doi: 10.1016/j.ejmech.2014.05.058. Epub 2014 May 24.
Eur J Med Chem. 2014.
PMID: 24915003
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Influence of the Dabcyl group on the cellular uptake of cationic peptides: short oligoarginines as efficient cell-penetrating peptides.
Szabó I, Illien F, Dókus LE, Yousef M, Baranyai Z, Bősze S, Ise S, Kawano K, Sagan S, Futaki S, Hudecz F, Bánóczi Z.
Szabó I, et al. Among authors: dokus le.
Amino Acids. 2021 Jul;53(7):1033-1049. doi: 10.1007/s00726-021-03003-w. Epub 2021 May 25.
Amino Acids. 2021.
PMID: 34032919
Free PMC article.
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Phage Display-Based Homing Peptide-Daunomycin Conjugates for Selective Drug Targeting to PANC-1 Pancreatic Cancer.
Dókus LE, Lajkó E, Ranđelović I, Mező D, Schlosser G, Kőhidai L, Tóvári J, Mező G.
Dókus LE, et al.
Pharmaceutics. 2020 Jun 22;12(6):576. doi: 10.3390/pharmaceutics12060576.
Pharmaceutics. 2020.
PMID: 32580307
Free PMC article.
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[Comparison of therapeutic peptides targeting pancreatic cancer].
Mezõ G, Dókus L, Schlosser G, Lajkó E, Szász Z, Ranđelović I, Biri-Kovács B, Tóvári J, Kõhidai L.
Mezõ G, et al.
Magy Onkol. 2019 Dec 9;63(4):301-308. Epub 2019 Oct 21.
Magy Onkol. 2019.
PMID: 31821385
Free article.
Hungarian.
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Energy-resolved HCD fragmentation of daunorubicin-peptide conjugates.
Al-Majidi M, Szabó D, Dókus L, Steckel A, Mező G, Schlosser G.
Al-Majidi M, et al.
J Mass Spectrom. 2020 Oct;55(10):e4641. doi: 10.1002/jms.4641.
J Mass Spectrom. 2020.
PMID: 32930447
No abstract available.
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