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Discovery of potent, orally bioavailable, small-molecule inhibitors of WNT signaling from a cell-based pathway screen.
J Med Chem. 2015 Feb 26;58(4):1717-35. doi: 10.1021/jm501436m. Epub 2015 Feb 13.
J Med Chem. 2015.
PMID: 25680029
Free PMC article.
Optimization of imidazo[4,5-b]pyridine-based kinase inhibitors: identification of a dual FLT3/Aurora kinase inhibitor as an orally bioavailable preclinical development candidate for the treatment of acute myeloid leukemia.
Bavetsias V, Crumpler S, Sun C, Avery S, Atrash B, Faisal A, Moore AS, Kosmopoulou M, Brown N, Sheldrake PW, Bush K, Henley A, Box G, Valenti M, de Haven Brandon A, Raynaud FI, Workman P, Eccles SA, Bayliss R, Linardopoulos S, Blagg J.
Bavetsias V, et al. Among authors: crumpler s.
J Med Chem. 2012 Oct 25;55(20):8721-34. doi: 10.1021/jm300952s. Epub 2012 Oct 8.
J Med Chem. 2012.
PMID: 23043539
Free PMC article.
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Discovery of Potent, Selective, and Orally Bioavailable Small-Molecule Modulators of the Mediator Complex-Associated Kinases CDK8 and CDK19.
Mallinger A, Schiemann K, Rink C, Stieber F, Calderini M, Crumpler S, Stubbs M, Adeniji-Popoola O, Poeschke O, Busch M, Czodrowski P, Musil D, Schwarz D, Ortiz-Ruiz MJ, Schneider R, Thai C, Valenti M, de Haven Brandon A, Burke R, Workman P, Dale T, Wienke D, Clarke PA, Esdar C, Raynaud FI, Eccles SA, Rohdich F, Blagg J.
Mallinger A, et al. Among authors: crumpler s.
J Med Chem. 2016 Feb 11;59(3):1078-101. doi: 10.1021/acs.jmedchem.5b01685. Epub 2016 Jan 21.
J Med Chem. 2016.
PMID: 26796641
Free PMC article.
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Aurora isoform selectivity: design and synthesis of imidazo[4,5-b]pyridine derivatives as highly selective inhibitors of Aurora-A kinase in cells.
Bavetsias V, Faisal A, Crumpler S, Brown N, Kosmopoulou M, Joshi A, Atrash B, Pérez-Fuertes Y, Schmitt JA, Boxall KJ, Burke R, Sun C, Avery S, Bush K, Henley A, Raynaud FI, Workman P, Bayliss R, Linardopoulos S, Blagg J.
Bavetsias V, et al. Among authors: crumpler s.
J Med Chem. 2013 Nov 27;56(22):9122-35. doi: 10.1021/jm401115g. Epub 2013 Nov 6.
J Med Chem. 2013.
PMID: 24195668
Free PMC article.
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Structural basis of poly(ADP-ribose) recognition by the multizinc binding domain of checkpoint with forkhead-associated and RING Domains (CHFR).
Oberoi J, Richards MW, Crumpler S, Brown N, Blagg J, Bayliss R.
Oberoi J, et al. Among authors: crumpler s.
J Biol Chem. 2010 Dec 10;285(50):39348-58. doi: 10.1074/jbc.M110.159855. Epub 2010 Sep 29.
J Biol Chem. 2010.
PMID: 20880844
Free PMC article.
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Responding to pulmonary-related blood transfusion reactions.
Bockhold C, Crumpler S.
Bockhold C, et al. Among authors: crumpler s.
Nursing. 2015 Sep;45(9):36-41; quiz 41-2. doi: 10.1097/01.NURSE.0000470412.33450.b1.
Nursing. 2015.
PMID: 26248201
Review.
No abstract available.
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