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Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins.
Science. 2015 Jun 5;348(6239):1106-12. doi: 10.1126/science.aaa4690.
Science. 2015.
PMID: 26045430
The antimalarial MMV688533 provides potential for single-dose cures with a high barrier to Plasmodium falciparum parasite resistance.
Murithi JM, Pascal C, Bath J, Boulenc X, Gnädig NF, Pasaje CFA, Rubiano K, Yeo T, Mok S, Klieber S, Desert P, Jiménez-Díaz MB, Marfurt J, Rouillier M, Cherkaoui-Rbati MH, Gobeau N, Wittlin S, Uhlemann AC, Price RN, Wirjanata G, Noviyanti R, Tumwebaze P, Cooper RA, Rosenthal PJ, Sanz LM, Gamo FJ, Joseph J, Singh S, Bashyam S, Augereau JM, Giraud E, Bozec T, Vermat T, Tuffal G, Guillon JM, Menegotto J, Sallé L, Louit G, Cabanis MJ, Nicolas MF, Doubovetzky M, Merino R, Bessila N, Angulo-Barturen I, Baud D, Bebrevska L, Escudié F, Niles JC, Blasco B, Campbell S, Courtemanche G, Fraisse L, Pellet A, Fidock DA, Leroy D.
Murithi JM, et al. Among authors: courtemanche g.
Sci Transl Med. 2021 Jul 21;13(603):eabg6013. doi: 10.1126/scitranslmed.abg6013.
Sci Transl Med. 2021.
PMID: 34290058
Free PMC article.
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Antitrypanosomal lead discovery: identification of a ligand-efficient inhibitor of Trypanosoma cruzi CYP51 and parasite growth.
Andriani G, Amata E, Beatty J, Clements Z, Coffey BJ, Courtemanche G, Devine W, Erath J, Juda CE, Wawrzak Z, Wood JT, Lepesheva GI, Rodriguez A, Pollastri MP.
Andriani G, et al. Among authors: courtemanche g.
J Med Chem. 2013 Mar 28;56(6):2556-67. doi: 10.1021/jm400012e. Epub 2013 Mar 13.
J Med Chem. 2013.
PMID: 23448316
Free PMC article.
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Metabolomics, lipidomics and proteomics profiling of myoblasts infected with Trypanosoma cruzi after treatment with different drugs against Chagas disease.
Hennig K, Abi-Ghanem J, Bunescu A, Meniche X, Biliaut E, Ouattara AD, Lewis MD, Kelly JM, Braillard S, Courtemanche G, Chatelain E, Béquet F.
Hennig K, et al. Among authors: courtemanche g.
Metabolomics. 2019 Aug 22;15(9):117. doi: 10.1007/s11306-019-1583-5.
Metabolomics. 2019.
PMID: 31440849
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Chagas Disease Drug Discovery: Multiparametric Lead Optimization against Trypanosoma cruzi in Acylaminobenzothiazole Series.
Fleau C, Padilla A, Miguel-Siles J, Quesada-Campos MT, Saiz-Nicolas I, Cotillo I, Cantizani Perez J, Tarleton RL, Marco M, Courtemanche G.
Fleau C, et al. Among authors: courtemanche g.
J Med Chem. 2019 Nov 27;62(22):10362-10375. doi: 10.1021/acs.jmedchem.9b01429. Epub 2019 Nov 18.
J Med Chem. 2019.
PMID: 31657555
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Activity in vivo of anti-Trypanosoma cruzi compounds selected from a high throughput screening.
Andriani G, Chessler AD, Courtemanche G, Burleigh BA, Rodriguez A.
Andriani G, et al. Among authors: courtemanche g.
PLoS Negl Trop Dis. 2011 Aug;5(8):e1298. doi: 10.1371/journal.pntd.0001298. Epub 2011 Aug 30.
PLoS Negl Trop Dis. 2011.
PMID: 21912715
Free PMC article.
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Bones of teleost fish demonstrate high fracture strain.
Fiedler IAK, Elmogazy O, Courtemanche G, Cardoso L, Berteau JP.
Fiedler IAK, et al. Among authors: courtemanche g.
J Biomech. 2021 May 7;120:110341. doi: 10.1016/j.jbiomech.2021.110341. Epub 2021 Mar 10.
J Biomech. 2021.
PMID: 33743397
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Zika antiviral chemotherapy: identification of drugs and promising starting points for drug discovery from an FDA-approved library.
Pascoalino BS, Courtemanche G, Cordeiro MT, Gil LH, Freitas-Junior L.
Pascoalino BS, et al. Among authors: courtemanche g.
F1000Res. 2016 Oct 14;5:2523. doi: 10.12688/f1000research.9648.1. eCollection 2016.
F1000Res. 2016.
PMID: 27909576
Free PMC article.
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