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Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds.
Borsari C, Santarem N, Torrado J, Olías AI, Corral MJ, Baptista C, Gul S, Wolf M, Kuzikov M, Ellinger B, Witt G, Gribbon P, Reinshagen J, Linciano P, Tait A, Costantino L, Freitas-Junior LH, Moraes CB, Bruno Dos Santos P, Alcântara LM, Franco CH, Bertolacini CD, Fontana V, Tejera Nevado P, Clos J, Alunda JM, Cordeiro-da-Silva A, Ferrari S, Costi MP. Borsari C, et al. Among authors: costi mp. Eur J Med Chem. 2017 Jan 27;126:1129-1135. doi: 10.1016/j.ejmech.2016.12.017. Epub 2016 Dec 9. Eur J Med Chem. 2017. PMID: 28064141
Update on antifolate drugs targets.
Costi MP, Ferrari S. Costi MP, et al. Curr Drug Targets. 2001 Jun;2(2):135-66. doi: 10.2174/1389450013348669. Curr Drug Targets. 2001. PMID: 11469716 Review.
Synthesis of N-(5,7-diamino-3-phenyl-quinoxalin-2-yl)-3,4,5-substituted anilines and N-[4[(5,7-diamino-3-phenylquinoxalin-2-yl)amino]benzoyl]-l-glutamic acid diethyl ester: evaluation of in vitro anti-cancer and anti-folate activities.
Corona P, Loriga M, Costi MP, Ferrari S, Paglietti G. Corona P, et al. Among authors: costi mp. Eur J Med Chem. 2008 Jan;43(1):189-203. doi: 10.1016/j.ejmech.2007.03.035. Epub 2007 Apr 18. Eur J Med Chem. 2008. PMID: 17532099
Discovery of potent pteridine reductase inhibitors to guide antiparasite drug development.
Cavazzuti A, Paglietti G, Hunter WN, Gamarro F, Piras S, Loriga M, Allecca S, Corona P, McLuskey K, Tulloch L, Gibellini F, Ferrari S, Costi MP. Cavazzuti A, et al. Among authors: costi mp. Proc Natl Acad Sci U S A. 2008 Feb 5;105(5):1448-53. doi: 10.1073/pnas.0704384105. Epub 2008 Feb 1. Proc Natl Acad Sci U S A. 2008. PMID: 18245389 Free PMC article.
137 results