Contino M - Search Results

1

Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A₁ Antagonists.

Val C, Rodríguez-García C, Prieto-Díaz R, Crespo A, Azuaje J, Carbajales C, Majellaro M, Díaz-Holguín A, Brea JM, Loza MI, Gioé-Gallo C, Contino M, Stefanachi A, García-Mera X, Estévez JC, Gutiérrez-de-Terán H, Sotelo E. Val C, et al. Among authors: contino m. J Med Chem. 2022 Feb 10;65(3):2091-2106. doi: 10.1021/acs.jmedchem.1c01636. Epub 2022 Jan 22. J Med Chem. 2022. PMID: 35068155 Free PMC article.

2

4-(tetralin-1-yl)- and 4-(naphthalen-1-yl)alkyl derivatives of 1-cyclohexylpiperazine as sigma receptor ligands with agonist sigma2 activity.

Berardi F, Ferorelli S, Abate C, Colabufo NA, Contino M, Perrone R, Tortorella V. Berardi F, et al. Among authors: contino m. J Med Chem. 2004 Apr 22;47(9):2308-17. doi: 10.1021/jm031026e. J Med Chem. 2004. PMID: 15084129

3

Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agents.

Leopoldo M, Berardi F, Colabufo NA, Contino M, Lacivita E, Niso M, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: contino m. J Med Chem. 2004 Dec 16;47(26):6616-24. doi: 10.1021/jm049702f. J Med Chem. 2004. PMID: 15588097

4

First structure-activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure.

Leopoldo M, Lacivita E, Colabufo NA, Contino M, Berardi F, Perrone R. Leopoldo M, et al. Among authors: contino m. J Med Chem. 2005 Dec 15;48(25):7919-22. doi: 10.1021/jm050729o. J Med Chem. 2005. PMID: 16335915

5

Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma(1) receptor.

Berardi F, Ferorelli S, Abate C, Pedone MP, Colabufo NA, Contino M, Perrone R. Berardi F, et al. Among authors: contino m. J Med Chem. 2005 Dec 29;48(26):8237-44. doi: 10.1021/jm050654o. J Med Chem. 2005. PMID: 16366605

6

Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides, a class of 5-HT7 receptor agents. 2.

Leopoldo M, Lacivita E, Contino M, Colabufo NA, Berardi F, Perrone R. Leopoldo M, et al. Among authors: contino m. J Med Chem. 2007 Aug 23;50(17):4214-21. doi: 10.1021/jm070487n. Epub 2007 Jul 25. J Med Chem. 2007. PMID: 17649988

7

Small P-gp modulating molecules: SAR studies on tetrahydroisoquinoline derivatives.

Colabufo NA, Berardi F, Cantore M, Perrone MG, Contino M, Inglese C, Niso M, Perrone R, Azzariti A, Simone GM, Porcelli L, Paradiso A. Colabufo NA, et al. Among authors: contino m. Bioorg Med Chem. 2008 Jan 1;16(1):362-73. doi: 10.1016/j.bmc.2007.09.039. Epub 2007 Sep 25. Bioorg Med Chem. 2008. PMID: 17936633

8

Tritium radiolabelling of PB28, a potent sigma-2 receptor ligand: pharmacokinetic and pharmacodynamic characterization.

Colabufo NA, Abate C, Contino M, Inglese C, Ferorelli S, Berardi F, Perrone R. Colabufo NA, et al. Among authors: contino m. Bioorg Med Chem Lett. 2008 Mar 15;18(6):2183-7. doi: 10.1016/j.bmcl.2007.12.056. Epub 2007 Dec 25. Bioorg Med Chem Lett. 2008. PMID: 18178434

9

4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators.

Colabufo NA, Berardi F, Cantore M, Perrone MG, Contino M, Inglese C, Niso M, Perrone R, Azzariti A, Simone GM, Paradiso A. Colabufo NA, et al. Among authors: contino m. Bioorg Med Chem. 2008 Apr 1;16(7):3732-43. doi: 10.1016/j.bmc.2008.01.055. Epub 2008 Feb 2. Bioorg Med Chem. 2008. PMID: 18276145

10

Structural modifications of N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides: influence on lipophilicity and 5-HT7 receptor activity. Part III.

Leopoldo M, Lacivita E, De Giorgio P, Fracasso C, Guzzetti S, Caccia S, Contino M, Colabufo NA, Berardi F, Perrone R. Leopoldo M, et al. Among authors: contino m. J Med Chem. 2008 Sep 25;51(18):5813-22. doi: 10.1021/jm800615e. J Med Chem. 2008. PMID: 18800769

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