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A nicotinamide phosphoribosyltransferase-GAPDH interaction sustains the stress-induced NMN/NAD+ salvage pathway in the nucleus.
Grolla AA, Miggiano R, Di Marino D, Bianchi M, Gori A, Orsomando G, Gaudino F, Galli U, Del Grosso E, Mazzola F, Angeletti C, Guarneri M, Torretta S, Calabrò M, Boumya S, Fan X, Colombo G, Travelli C, Rocchio F, Aronica E, Wohlschlegel JA, Deaglio S, Rizzi M, Genazzani AA, Garavaglia S. Grolla AA, et al. Among authors: colombo g. J Biol Chem. 2020 Mar 13;295(11):3635-3651. doi: 10.1074/jbc.RA119.010571. Epub 2020 Jan 27. J Biol Chem. 2020. PMID: 31988240 Free PMC article.
NAMPT: A pleiotropic modulator of monocytes and macrophages.
Travelli C, Colombo G, Mola S, Genazzani AA, Porta C. Travelli C, et al. Among authors: colombo g. Pharmacol Res. 2018 Sep;135:25-36. doi: 10.1016/j.phrs.2018.06.022. Epub 2018 Jul 18. Pharmacol Res. 2018. PMID: 30031171 Review.
Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group.
Travelli C, Aprile S, Mattoteia D, Colombo G, Clemente N, Scanziani E, Terrazzino S, Alisi MA, Polenzani L, Grosa G, Genazzani AA, Tron GC, Galli U. Travelli C, et al. Among authors: colombo g. Eur J Med Chem. 2019 Nov 1;181:111576. doi: 10.1016/j.ejmech.2019.111576. Epub 2019 Aug 1. Eur J Med Chem. 2019. PMID: 31400709
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic Activity.
Serafini M, Torre E, Aprile S, Grosso ED, Gesù A, Griglio A, Colombo G, Travelli C, Paiella S, Adamo A, Orecchini E, Coletti A, Pallotta MT, Ugel S, Massarotti A, Pirali T, Fallarini S. Serafini M, et al. Among authors: colombo g. J Med Chem. 2020 Mar 26;63(6):3047-3065. doi: 10.1021/acs.jmedchem.9b01809. Epub 2020 Mar 17. J Med Chem. 2020. PMID: 32150677
Neutralization of extracellular NAMPT (nicotinamide phosphoribosyltransferase) ameliorates experimental murine colitis.
Colombo G, Clemente N, Zito A, Bracci C, Colombo FS, Sangaletti S, Jachetti E, Ribaldone DG, Caviglia GP, Pastorelli L, De Andrea M, Naviglio S, Lucafò M, Stocco G, Grolla AA, Campolo M, Casili G, Cuzzocrea S, Esposito E, Malavasi F, Genazzani AA, Porta C, Travelli C. Colombo G, et al. Among authors: colombo fs. J Mol Med (Berl). 2020 Apr;98(4):595-612. doi: 10.1007/s00109-020-01892-0. Epub 2020 Apr 27. J Mol Med (Berl). 2020. PMID: 32338310 Free article.
Recent Advances in NAMPT Inhibitors: A Novel Immunotherapic Strategy.
Galli U, Colombo G, Travelli C, Tron GC, Genazzani AA, Grolla AA. Galli U, et al. Among authors: colombo g. Front Pharmacol. 2020 May 12;11:656. doi: 10.3389/fphar.2020.00656. eCollection 2020. Front Pharmacol. 2020. PMID: 32477131 Free PMC article. Review.
1,367 results