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IMI European Lead Factory - democratizing access to high-throughput screening.
Jones PS, Boucharens S, McElroy SP, Morrison A, Honarnejad S, van Boeckel S, van den Hurk H, Basting D, Hüser J, Jaroch S, Ottow E, Benningshof J, Folmer RHA, Leemhuis F, Kramer-Verhulst PM, Nies VJM, Orrling KM, Rijnders T, Pfander C, Engkvist O, Pairaudeau G, Simpson PB, Ortholand JY, Roche D, Dömling A, Kühnert SM, Roevens PWM, van Vlijmen H, van Wanrooij EJA, Verbruggen C, Nussbaumer P, Ovaa H, van der Stelt M, Simonsen KB, Tagmose L, Waldmann H, Duffy J, Finsinger D, Jurzak M, Burgess-Brown NA, Lee WH, Rutjes FPJT, Haag H, Kallus C, Mors H, Dorval T, Lesur B, Ramon Olayo F, Hamza D, Jones G, Pearce C, Piechot A, Tzalis D, Clausen MH, Davis J, Derouane D, Vermeiren C, Kaiser M, Stockman RA, Barrault DV, Pannifer AD, Swedlow JR, Nelson AS, Orru RVA, Ruijter E, van Helden SP, Li VM, Vries T, de Vlieger JSB. Jones PS, et al. Among authors: clausen mh. Nat Rev Drug Discov. 2022 Apr;21(4):245-246. doi: 10.1038/d41573-021-00196-3. Nat Rev Drug Discov. 2022. PMID: 34907316 No abstract available.
Synthesis of 1,4,5 trisubstituted γ-lactams via a 3-component cascade reaction.
Petersen MÅ, Mortensen MA, Cohrt AE, Petersen R, Wu P, Fleury-Brégeot N, Morgentin R, Lardy C, Nielsen TE, Clausen MH. Petersen MÅ, et al. Among authors: clausen mh. Bioorg Med Chem. 2015 Jun 1;23(11):2695-8. doi: 10.1016/j.bmc.2015.01.041. Epub 2015 Jan 31. Bioorg Med Chem. 2015. PMID: 25684425
Synthesis of branched and linear 1,4-linked galactan oligosaccharides.
Andersen MCF, Boos I, Kinnaert C, Awan SI, Pedersen HL, Kračun SK, Lanz G, Rydahl MG, Kjærulff L, Håkansson M, Kimbung R, Logan DT, Gotfredsen CH, Willats WGT, Clausen MH. Andersen MCF, et al. Among authors: clausen mh. Org Biomol Chem. 2018 Feb 14;16(7):1157-1162. doi: 10.1039/c7ob03035e. Org Biomol Chem. 2018. PMID: 29367995
The 3F Library: Fluorinated Fsp3 -Rich Fragments for Expeditious 19 F NMR Based Screening.
Troelsen NS, Shanina E, Gonzalez-Romero D, Danková D, Jensen ISA, Śniady KJ, Nami F, Zhang H, Rademacher C, Cuenda A, Gotfredsen CH, Clausen MH. Troelsen NS, et al. Among authors: clausen mh. Angew Chem Int Ed Engl. 2020 Feb 3;59(6):2204-2210. doi: 10.1002/anie.201913125. Epub 2019 Dec 17. Angew Chem Int Ed Engl. 2020. PMID: 31724281
Azodyrecins A-C: Azoxides from a Soil-Derived Streptomyces Species.
Wibowo M, Gotfredsen CH, Sassetti E, Melchiorsen J, Clausen MH, Gram L, Ding L. Wibowo M, et al. Among authors: clausen mh. J Nat Prod. 2020 Dec 24;83(12):3519-3525. doi: 10.1021/acs.jnatprod.0c00339. Epub 2020 Nov 20. J Nat Prod. 2020. PMID: 33216557
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