Discovery and optimization of selective RET inhibitors via scaffold hopping.
Luo Z, Wang L, Fu Z, Shuai B, Luo M, Hu G, Chen J, Sun J, Wang J, Li J, Chen S, Zhang Y.
Luo Z, et al. Among authors: chen j, chen s.
Bioorg Med Chem Lett. 2021 Sep 1;47:128149. doi: 10.1016/j.bmcl.2021.128149. Epub 2021 May 28.
Bioorg Med Chem Lett. 2021.
PMID: 34058344