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CCR9 Antagonists in the Treatment of Ulcerative Colitis.
Mediators Inflamm. 2015;2015:628340. doi: 10.1155/2015/628340. Epub 2015 Sep 20.
Mediators Inflamm. 2015.
PMID: 26457007
Free PMC article.
A systemically-administered small molecule antagonist of CCR9 acts as a tissue-selective inhibitor of lymphocyte trafficking.
Tubo NJ, Wurbel MA, Charvat TT, Schall TJ, Walters MJ, Campbell JJ.
Tubo NJ, et al. Among authors: charvat tt.
PLoS One. 2012;7(11):e50498. doi: 10.1371/journal.pone.0050498. Epub 2012 Nov 29.
PLoS One. 2012.
PMID: 23209760
Free PMC article.
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The adipokine chemerin amplifies electrical field-stimulated contraction in the isolated rat superior mesenteric artery.
Darios ES, Winner BM, Charvat T, Krasinksi A, Punna S, Watts SW.
Darios ES, et al.
Am J Physiol Heart Circ Physiol. 2016 Aug 1;311(2):H498-507. doi: 10.1152/ajpheart.00998.2015. Epub 2016 Jul 1.
Am J Physiol Heart Circ Physiol. 2016.
PMID: 27371688
Free PMC article.
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Abrogation of CC chemokine receptor 9 ameliorates collagen-induced arthritis of mice.
Yokoyama W, Kohsaka H, Kaneko K, Walters M, Takayasu A, Fukuda S, Miyabe C, Miyabe Y, Love PE, Nakamoto N, Kanai T, Watanabe-Imai K, Charvat TT, Penfold ME, Jaen J, Schall TJ, Harigai M, Miyasaka N, Nanki T.
Yokoyama W, et al. Among authors: charvat tt.
Arthritis Res Ther. 2014 Sep 24;16(5):445. doi: 10.1186/s13075-014-0445-9.
Arthritis Res Ther. 2014.
PMID: 25248373
Free PMC article.
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1-(4-Phenylpiperazin-1-yl)-2-(1H-pyrazol-1-yl)ethanones as novel CCR1 antagonists.
Pennell AM, Aggen JB, Sen S, Chen W, Xu Y, Sullivan E, Li L, Greenman K, Charvat T, Hansen D, Dairaghi DJ, Wright JJ, Zhang P.
Pennell AM, et al.
Bioorg Med Chem Lett. 2013 Mar 1;23(5):1228-31. doi: 10.1016/j.bmcl.2013.01.005. Epub 2013 Jan 11.
Bioorg Med Chem Lett. 2013.
PMID: 23374868
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Chemerin connects fat to arterial contraction.
Watts SW, Dorrance AM, Penfold ME, Rourke JL, Sinal CJ, Seitz B, Sullivan TJ, Charvat TT, Thompson JM, Burnett R, Fink GD.
Watts SW, et al. Among authors: charvat tt.
Arterioscler Thromb Vasc Biol. 2013 Jun;33(6):1320-8. doi: 10.1161/ATVBAHA.113.301476. Epub 2013 Apr 4.
Arterioscler Thromb Vasc Biol. 2013.
PMID: 23559624
Free PMC article.
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Increased expression of chemerin in squamous esophageal cancer myofibroblasts and role in recruitment of mesenchymal stromal cells.
Kumar JD, Holmberg C, Kandola S, Steele I, Hegyi P, Tiszlavicz L, Jenkins R, Beynon RJ, Peeney D, Giger OT, Alqahtani A, Wang TC, Charvat TT, Penfold M, Dockray GJ, Varro A.
Kumar JD, et al. Among authors: charvat tt.
PLoS One. 2014 Aug 15;9(7):e104877. doi: 10.1371/journal.pone.0104877. eCollection 2014.
PLoS One. 2014.
PMID: 25127029
Free PMC article.
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Design, synthesis, and biological evaluation of chicoric acid analogs as inhibitors of HIV-1 integrase.
Charvat TT, Lee DJ, Robinson WE, Chamberlin AR.
Charvat TT, et al.
Bioorg Med Chem. 2006 Jul 1;14(13):4552-67. doi: 10.1016/j.bmc.2006.02.030. Epub 2006 Mar 9.
Bioorg Med Chem. 2006.
PMID: 16524737
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