Benzo[b]thiophene-2-carboxamides as novel opioid receptor agonists with potent analgesic effect and reduced constipation.
Kuppusamy R, Hsu YT, Ke YY, Chang PW, Chang YC, Chang HF, Wang PC, Lin YH, Huang YC, Yeh TK, Chuang JY, Loh HH, Shih C, Chen CT, Yeh SH, Ueng SH.
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Eur J Med Chem. 2022 Dec 5;243:114728. doi: 10.1016/j.ejmech.2022.114728. Epub 2022 Aug 31.
Eur J Med Chem. 2022.
PMID: 36084534