Chaiken I - Search Results

1

HIV-1 Env-Dependent Cell Killing by Bifunctional Small-Molecule/Peptide Conjugates.

Gaffney A, Nangarlia A, Ang CG, Gossert S, Rashad Ahmed AA, Hossain MA, Abrams CF, Smith AB 3rd, Chaiken I. Gaffney A, et al. Among authors: chaiken i. ACS Chem Biol. 2021 Jan 15;16(1):193-204. doi: 10.1021/acschembio.0c00888. Epub 2021 Jan 7. ACS Chem Biol. 2021. PMID: 33410670 Free PMC article.

2

From receptor recognition mechanisms to bioinspired mimetic antagonists in HIV-1/cell docking.

Dowd CS, Zhang W, Li C, Chaiken IM. Dowd CS, et al. Among authors: chaiken im. J Chromatogr B Biomed Sci Appl. 2001 Apr 5;753(2):327-35. doi: 10.1016/s0378-4347(00)00567-3. J Chromatogr B Biomed Sci Appl. 2001. PMID: 11334348 Review.

3

Beta-turn Phe in HIV-1 Env binding site of CD4 and CD4 mimetic miniprotein enhances Env binding affinity but is not required for activation of co-receptor/17b site.

Dowd CS, Leavitt S, Babcock G, Godillot AP, Van Ryk D, Canziani GA, Sodroski J, Freire E, Chaiken IM. Dowd CS, et al. Biochemistry. 2002 Jun 4;41(22):7038-46. doi: 10.1021/bi012168i. Biochemistry. 2002. PMID: 12033937

4

Peptide-small molecule hybrids via orthogonal deprotection-chemoselective conjugation to cysteine-anchored scaffolds. A model study.

Smith AB 3rd, Savinov SN, Manjappara UV, Chaiken IM. Smith AB 3rd, et al. Org Lett. 2002 Nov 14;4(23):4041-4. doi: 10.1021/ol026736d. Org Lett. 2002. PMID: 12423081

5

Salivary agglutinin inhibits HIV type 1 infectivity through interaction with viral glycoprotein 120.

Wu Z, Van Ryk D, Davis C, Abrams WR, Chaiken I, Magnani J, Malamud D. Wu Z, et al. Among authors: chaiken i. AIDS Res Hum Retroviruses. 2003 Mar;19(3):201-9. doi: 10.1089/088922203763315704. AIDS Res Hum Retroviruses. 2003. PMID: 12689412

6

Mode of action for linear peptide inhibitors of HIV-1 gp120 interactions.

Biorn AC, Cocklin S, Madani N, Si Z, Ivanovic T, Samanen J, Van Ryk DI, Pantophlet R, Burton DR, Freire E, Sodroski J, Chaiken IM. Biorn AC, et al. Among authors: chaiken im. Biochemistry. 2004 Feb 24;43(7):1928-38. doi: 10.1021/bi035088i. Biochemistry. 2004. PMID: 14967033

7

Small-molecule inhibitors of HIV-1 entry block receptor-induced conformational changes in the viral envelope glycoproteins.

Si Z, Madani N, Cox JM, Chruma JJ, Klein JC, Schön A, Phan N, Wang L, Biorn AC, Cocklin S, Chaiken I, Freire E, Smith AB 3rd, Sodroski JG. Si Z, et al. Among authors: chaiken i. Proc Natl Acad Sci U S A. 2004 Apr 6;101(14):5036-41. doi: 10.1073/pnas.0307953101. Epub 2004 Mar 29. Proc Natl Acad Sci U S A. 2004. PMID: 15051887 Free PMC article.

8

Structural determinants for affinity enhancement of a dual antagonist peptide entry inhibitor of human immunodeficiency virus type-1.

Gopi H, Umashankara M, Pirrone V, LaLonde J, Madani N, Tuzer F, Baxter S, Zentner I, Cocklin S, Jawanda N, Miller SR, Schön A, Klein JC, Freire E, Krebs FC, Smith AB, Sodroski J, Chaiken I. Gopi H, et al. Among authors: chaiken i. J Med Chem. 2008 May 8;51(9):2638-47. doi: 10.1021/jm070814r. Epub 2008 Apr 11. J Med Chem. 2008. PMID: 18402432 Free PMC article.

9

Introducing metallocene into a triazole peptide conjugate reduces its off-rate and enhances its affinity and antiviral potency for HIV-1 gp120.

Gopi H, Cocklin S, Pirrone V, McFadden K, Tuzer F, Zentner I, Ajith S, Baxter S, Jawanda N, Krebs FC, Chaiken IM. Gopi H, et al. Among authors: chaiken im. J Mol Recognit. 2009 Mar-Apr;22(2):169-74. doi: 10.1002/jmr.892. J Mol Recognit. 2009. PMID: 18498083 Free PMC article.

10

Use of the quartz crystal microbalance to monitor ligand-induced conformational rearrangements in HIV-1 envelope protein gp120.

Lee HS, Contarino M, Umashankara M, Schön A, Freire E, Smith AB 3rd, Chaiken IM, Penn LS. Lee HS, et al. Anal Bioanal Chem. 2010 Feb;396(3):1143-52. doi: 10.1007/s00216-009-3313-8. Epub 2009 Dec 17. Anal Bioanal Chem. 2010. PMID: 20016882 Free PMC article.

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