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A Novel MYCN-Specific Antigene Oligonucleotide Deregulates Mitochondria and Inhibits Tumor Growth in MYCN-Amplified Neuroblastoma.
Cancer Res. 2019 Dec 15;79(24):6166-6177. doi: 10.1158/0008-5472.CAN-19-0008. Epub 2019 Oct 15.
Cancer Res. 2019.
PMID: 31615807
The MYCN inhibitor BGA002 restores the retinoic acid response leading to differentiation or apoptosis by the mTOR block in MYCN-amplified neuroblastoma.
Lampis S, Raieli S, Montemurro L, Bartolucci D, Amadesi C, Bortolotti S, Angelucci S, Scardovi AL, Nieddu G, Cerisoli L, Paganelli F, Valente S, Fischer M, Martelli AM, Pasquinelli G, Pession A, Hrelia P, Tonelli R.
Lampis S, et al. Among authors: cerisoli l.
J Exp Clin Cancer Res. 2022 Apr 30;41(1):160. doi: 10.1186/s13046-022-02367-5.
J Exp Clin Cancer Res. 2022.
PMID: 35490242
Free PMC article.
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Antigene MYCN Silencing by BGA002 Inhibits SCLC Progression Blocking mTOR Pathway and Overcomes Multidrug Resistance.
Bortolotti S, Angelucci S, Montemurro L, Bartolucci D, Raieli S, Lampis S, Amadesi C, Scardovi A, Nieddu G, Cerisoli L, Paganelli F, Chiarini F, Teti G, Falconi M, Pession A, Hrelia P, Tonelli R.
Bortolotti S, et al. Among authors: cerisoli l.
Cancers (Basel). 2023 Feb 3;15(3):990. doi: 10.3390/cancers15030990.
Cancers (Basel). 2023.
PMID: 36765949
Free PMC article.
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Novel insights into the chemistry of an old medicine: A general degradative pathway for penicillins from a piperacillin/tazobactam stability study.
Viola A, Ferrazzano L, Martelli G, Cerisoli L, Ricci A, Tolomelli A, Cabri W.
Viola A, et al. Among authors: cerisoli l.
Eur J Pharm Sci. 2019 Aug 1;136:104957. doi: 10.1016/j.ejps.2019.104957. Epub 2019 Jun 14.
Eur J Pharm Sci. 2019.
PMID: 31202896
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The First Enantioselective Organocatalytic Synthesis of 3-Spiro-α-Alkylidene-γ-Butyrolactone Oxindoles.
Cerisoli L, Lombardo M, Trombini C, Quintavalla A.
Cerisoli L, et al.
Chemistry. 2016 Mar 7;22(11):3865-72. doi: 10.1002/chem.201504157. Epub 2016 Jan 7.
Chemistry. 2016.
PMID: 26743560
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Pyrrole macrocyclic ligands for Cu-catalyzed asymmetric Henry reactions.
Gualandi A, Cerisoli L, Stoeckli-Evans H, Savoia D.
Gualandi A, et al. Among authors: cerisoli l.
J Org Chem. 2011 May 6;76(9):3399-408. doi: 10.1021/jo200318b. Epub 2011 Apr 6.
J Org Chem. 2011.
PMID: 21417436
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Chemical modifications designed to improve peptide stability: incorporation of non-natural amino acids, pseudo-peptide bonds, and cyclization.
Gentilucci L, De Marco R, Cerisoli L.
Gentilucci L, et al. Among authors: cerisoli l.
Curr Pharm Des. 2010;16(28):3185-203. doi: 10.2174/138161210793292555.
Curr Pharm Des. 2010.
PMID: 20687878
Review.
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