Skip to main page content
U.S. flag

An official website of the United States government

Dot gov

The .gov means it’s official.
Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you’re on a federal government site.

Https

The site is secure.
The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.

Access keys NCBI Homepage MyNCBI Homepage Main Content Main Navigation

Search Page

Filters

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

Search Results

16 results

Filters applied: . Clear all
Results are displayed in a computed author sort order. The Results By Year timeline is not available.
Page 1
New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains.
Felicetti T, Cedraro N, Astolfi A, Cernicchi G, Mangiaterra G, Vaiasicca S, Massari S, Manfroni G, Barreca ML, Tabarrini O, Biavasco F, Cecchetti V, Vignaroli C, Sabatini S. Felicetti T, et al. Among authors: cedraro n. Eur J Med Chem. 2022 Nov 5;241:114656. doi: 10.1016/j.ejmech.2022.114656. Epub 2022 Aug 6. Eur J Med Chem. 2022. PMID: 35963131
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors.
Felicetti T, Mangiaterra G, Cannalire R, Cedraro N, Pietrella D, Astolfi A, Massari S, Tabarrini O, Manfroni G, Barreca ML, Cecchetti V, Biavasco F, Sabatini S. Felicetti T, et al. Among authors: cedraro n. J Enzyme Inhib Med Chem. 2020 Dec;35(1):584-597. doi: 10.1080/14756366.2020.1719083. J Enzyme Inhib Med Chem. 2020. PMID: 31992093 Free PMC article.
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search.
Cedraro N, Cannalire R, Astolfi A, Mangiaterra G, Felicetti T, Vaiasicca S, Cernicchi G, Massari S, Manfroni G, Tabarrini O, Cecchetti V, Barreca ML, Biavasco F, Sabatini S. Cedraro N, et al. ChemMedChem. 2021 Oct 6;16(19):3044-3059. doi: 10.1002/cmdc.202100282. Epub 2021 Jun 26. ChemMedChem. 2021. PMID: 34032014 Free PMC article.
16 results