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Side-Chain Modified Ergosterol and Stigmasterol Derivatives as Liver X Receptor Agonists.
J Med Chem. 2017 Aug 10;60(15):6548-6562. doi: 10.1021/acs.jmedchem.7b00091. Epub 2017 Jul 25.
J Med Chem. 2017.
PMID: 28741954
C24-hydroxylated stigmastane derivatives as Liver X Receptor agonists.
Castro Navas FF, Giorgi G, Maggioni D, Pacciarini M, Russo V, Marinozzi M.
Castro Navas FF, et al.
Chem Phys Lipids. 2018 May;212:44-50. doi: 10.1016/j.chemphyslip.2018.01.005. Epub 2018 Jan 17.
Chem Phys Lipids. 2018.
PMID: 29352964
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Synthesis, biological evaluation, in silico modeling and crystallization of novel small monocationic molecules with potent antiproliferative activity by dual mechanism.
Serrán-Aguilera L, Mariotto E, Rubbini G, Castro Navas FF, Marco C, Carrasco-Jiménez MP, Ballarotto M, Macchiarulo A, Hurtado-Guerrero R, Viola G, Lopez-Cara LC.
Serrán-Aguilera L, et al. Among authors: castro navas ff.
Eur J Med Chem. 2020 Dec 1;207:112797. doi: 10.1016/j.ejmech.2020.112797. Epub 2020 Sep 6.
Eur J Med Chem. 2020.
PMID: 32977218
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New more polar symmetrical bipyridinic compounds: new strategy for the inhibition of choline kinase α1.
Castro-Navas FF, Schiaffino-Ortega S, Carrasco-Jimenez MP, Ríos-Marco P, Marco C, Espinosa A, Gallo MA, Mariotto E, Basso G, Viola G, Entrena-Guadix A, López-Cara LC.
Castro-Navas FF, et al.
Future Med Chem. 2015;7(4):417-36. doi: 10.4155/fmc.15.1.
Future Med Chem. 2015.
PMID: 25875870
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