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Multivalent supramolecular dendrimer-based drugs.
Galeazzi S, Hermans TM, Paolino M, Anzini M, Mennuni L, Giordani A, Caselli G, Makovec F, Meijer EW, Vomero S, Cappelli A. Galeazzi S, et al. Among authors: cappelli a. Biomacromolecules. 2010 Jan 11;11(1):182-6. doi: 10.1021/bm901055a. Biomacromolecules. 2010. PMID: 19957993
Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold.
Castriconi F, Paolino M, Giuliani G, Anzini M, Campiani G, Mennuni L, Sabatini C, Lanza M, Caselli G, De Rienzo F, Menziani MC, Sbraccia M, Molinari P, Costa T, Cappelli A. Castriconi F, et al. Among authors: cappelli a. Eur J Med Chem. 2014 Jul 23;82:36-46. doi: 10.1016/j.ejmech.2014.05.015. Epub 2014 May 5. Eur J Med Chem. 2014. PMID: 24871995
Dendrimeric tetravalent ligands for the serotonin-gated ion channel.
Paolino M, Mennuni L, Giuliani G, Anzini M, Lanza M, Caselli G, Galimberti C, Menziani MC, Donati A, Cappelli A. Paolino M, et al. Among authors: cappelli a. Chem Commun (Camb). 2014 Aug 11;50(62):8582-5. doi: 10.1039/c4cc02502d. Epub 2014 Jun 23. Chem Commun (Camb). 2014. PMID: 24956157
Supramolecular glycodendrimer-based hybrid drugs.
Paolino M, Komber H, Mennuni L, Caselli G, Appelhans D, Voit B, Cappelli A. Paolino M, et al. Among authors: cappelli a. Biomacromolecules. 2014 Nov 10;15(11):3985-93. doi: 10.1021/bm501057d. Epub 2014 Oct 20. Biomacromolecules. 2014. PMID: 25286342
Design, Synthesis, and Biological Evaluation of Imidazo[1,5-a]quinoline as Highly Potent Ligands of Central Benzodiazepine Receptors.
Cappelli A, Anzini M, Castriconi F, Grisci G, Paolino M, Braile C, Valenti S, Giuliani G, Vomero S, Di Capua A, Betti L, Giannaccini G, Lucacchini A, Ghelardini C, Di Cesare Mannelli L, Frosini M, Ricci L, Giorgi G, Mascia MP, Biggio G. Cappelli A, et al. J Med Chem. 2016 Apr 14;59(7):3353-72. doi: 10.1021/acs.jmedchem.6b00034. Epub 2016 Mar 24. J Med Chem. 2016. PMID: 26982523
362 results