Canale V - Search Results

1

A dual-acting 5-HT₆ receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties.

Canale V, Grychowska K, Kurczab R, Ryng M, Keeri AR, Satała G, Olejarz-Maciej A, Koczurkiewicz P, Drop M, Blicharz K, Piska K, Pękala E, Janiszewska P, Krawczyk M, Walczak M, Chaumont-Dubel S, Bojarski AJ, Marin P, Popik P, Zajdel P. Canale V, et al. Eur J Med Chem. 2020 Dec 15;208:112765. doi: 10.1016/j.ejmech.2020.112765. Epub 2020 Aug 22. Eur J Med Chem. 2020. PMID: 32949963

2

Quinolinesulfonamides of aryloxy-/arylthio-ethyl piperidines: influence of an arylether fragment on 5-HT1A/5-HT7 receptor selectivity.

Grychowska K, Marciniec K, Canale V, Szymiec M, Glanowski G, Satała G, Maślankiewicz A, Pawłowski M, Bojarski AJ, Zajdel P. Grychowska K, et al. Among authors: canale v. Arch Pharm (Weinheim). 2013 Mar;346(3):180-8. doi: 10.1002/ardp.201200322. Epub 2013 Feb 4. Arch Pharm (Weinheim). 2013. PMID: 23381952

3

Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT(7) and 5-HT(1A) receptor ligands.

Canale V, Guzik P, Kurczab R, Verdie P, Satała G, Kubica B, Pawłowski M, Martinez J, Subra G, Bojarski AJ, Zajdel P. Canale V, et al. Eur J Med Chem. 2014 May 6;78:10-22. doi: 10.1016/j.ejmech.2014.03.005. Epub 2014 Mar 5. Eur J Med Chem. 2014. PMID: 24675176

4

Towards novel 5-HT7versus 5-HT1A receptor ligands among LCAPs with cyclic amino acid amide fragments: design, synthesis, and antidepressant properties. Part II.

Canale V, Kurczab R, Partyka A, Satała G, Witek J, Jastrzębska-Więsek M, Pawłowski M, Bojarski AJ, Wesołowska A, Zajdel P. Canale V, et al. Eur J Med Chem. 2015 Mar 6;92:202-11. doi: 10.1016/j.ejmech.2014.12.041. Epub 2014 Dec 24. Eur J Med Chem. 2015. PMID: 25555143

5

Preliminary mutagenicity and genotoxicity evaluation of selected arylsulfonamide derivatives of (aryloxy)alkylamines with potential psychotropic properties.

Powroźnik B, Słoczyńska K, Canale V, Grychowska K, Zajdel P, Pękala E. Powroźnik B, et al. Among authors: canale v. J Appl Genet. 2016 May;57(2):263-70. doi: 10.1007/s13353-015-0322-5. Epub 2015 Oct 6. J Appl Genet. 2016. PMID: 26440375

6

Towards new 5-HT7 antagonists among arylsulfonamide derivatives of (aryloxy)ethyl-alkyl amines: Multiobjective based design, synthesis, and antidepressant and anxiolytic properties.

Canale V, Kurczab R, Partyka A, Satała G, Lenda T, Jastrzębska-Więsek M, Wesołowska A, Bojarski AJ, Zajdel P. Canale V, et al. Eur J Med Chem. 2016 Jan 27;108:334-346. doi: 10.1016/j.ejmech.2015.11.040. Epub 2015 Nov 30. Eur J Med Chem. 2016. PMID: 26698537

7

N-Alkylated arylsulfonamides of (aryloxy)ethyl piperidines: 5-HT(7) receptor selectivity versus multireceptor profile.

Canale V, Kurczab R, Partyka A, Satała G, Słoczyńska K, Kos T, Jastrzębska-Więsek M, Siwek A, Pękala E, Bojarski AJ, Wesołowska A, Popik P, Zajdel P. Canale V, et al. Bioorg Med Chem. 2016 Jan 15;24(2):130-9. doi: 10.1016/j.bmc.2015.11.041. Epub 2015 Nov 30. Bioorg Med Chem. 2016. PMID: 26706111

8

An Algorithm to Identify Target-Selective Ligands - A Case Study of 5-HT7/5-HT1A Receptor Selectivity.

Kurczab R, Canale V, Zajdel P, Bojarski AJ. Kurczab R, et al. Among authors: canale v. PLoS One. 2016 Jun 7;11(6):e0156986. doi: 10.1371/journal.pone.0156986. eCollection 2016. PLoS One. 2016. PMID: 27271158 Free PMC article.

9

N1-Azinylsulfonyl-1H-indoles: 5-HT6 Receptor Antagonists with Procognitive and Antidepressant-Like Properties.

Zajdel P, Marciniec K, Satała G, Canale V, Kos T, Partyka A, Jastrzębska-Więsek M, Wesołowska A, Basińska-Ziobroń A, Wójcikowski J, Daniel WA, Bojarski AJ, Popik P. Zajdel P, et al. Among authors: canale v. ACS Med Chem Lett. 2016 Apr 7;7(6):618-22. doi: 10.1021/acsmedchemlett.6b00056. eCollection 2016 Jun 9. ACS Med Chem Lett. 2016. PMID: 27326337 Free PMC article.

10

Arylsulfonamide derivatives of (aryloxy)ethyl pyrrolidines and piperidines as α₁-adrenergic receptor antagonist with uro-selective activity.

Rak A, Canale V, Marciniec K, Żmudzki P, Kotańska M, Knutelska J, Siwek A, Stachowicz G, Bednarski M, Nowiński L, Zygmunt M, Zajdel P, Sapa J. Rak A, et al. Among authors: canale v. Bioorg Med Chem. 2016 Nov 1;24(21):5582-5591. doi: 10.1016/j.bmc.2016.09.017. Epub 2016 Sep 10. Bioorg Med Chem. 2016. PMID: 27658792

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