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Anti-Inflammatory, Antioxidant, and WAT/BAT-Conversion Stimulation Induced by Novel PPAR Ligands: Results from Ex Vivo and In Vitro Studies.
Recinella L, De Filippis B, Libero ML, Ammazzalorso A, Chiavaroli A, Orlando G, Ferrante C, Giampietro L, Veschi S, Cama A, Mannino F, Gasparo I, Bitto A, Amoroso R, Brunetti L, Leone S. Recinella L, et al. Among authors: cama a. Pharmaceuticals (Basel). 2023 Feb 24;16(3):346. doi: 10.3390/ph16030346. Pharmaceuticals (Basel). 2023. PMID: 36986448 Free PMC article.
Anti-Inflammatory and Antioxidant Effects Induced by Allium sativum L. Extracts on an Ex Vivo Experimental Model of Ulcerative Colitis.
Recinella L, Gorica E, Chiavaroli A, Fraschetti C, Filippi A, Cesa S, Cairone F, Martelli A, Calderone V, Veschi S, Lanuti P, Cama A, Orlando G, Ferrante C, Menghini L, Di Simone SC, Acquaviva A, Libero ML, Nilofar, Brunetti L, Leone S. Recinella L, et al. Among authors: cama a. Foods. 2022 Nov 9;11(22):3559. doi: 10.3390/foods11223559. Foods. 2022. PMID: 36429152 Free PMC article.
Novel Phenyldiazenyl Fibrate Analogues as PPAR α/γ/δ Pan-Agonists for the Amelioration of Metabolic Syndrome.
Giampietro L, Laghezza A, Cerchia C, Florio R, Recinella L, Capone F, Ammazzalorso A, Bruno I, De Filippis B, Fantacuzzi M, Ferrante C, Maccallini C, Tortorella P, Verginelli F, Brunetti L, Cama A, Amoroso R, Loiodice F, Lavecchia A. Giampietro L, et al. Among authors: cama a. ACS Med Chem Lett. 2019 Feb 25;10(4):545-551. doi: 10.1021/acsmedchemlett.8b00574. eCollection 2019 Apr 11. ACS Med Chem Lett. 2019. PMID: 30996794 Free PMC article.
Synthesis of novel benzothiazole amides: Evaluation of PPAR activity and anti-proliferative effects in paraganglioma, pancreatic and colorectal cancer cell lines.
Ammazzalorso A, De Lellis L, Florio R, Laghezza A, De Filippis B, Fantacuzzi M, Giampietro L, Maccallini C, Tortorella P, Veschi S, Loiodice F, Cama A, Amoroso R. Ammazzalorso A, et al. Among authors: cama a. Bioorg Med Chem Lett. 2019 Aug 15;29(16):2302-2306. doi: 10.1016/j.bmcl.2019.06.020. Epub 2019 Jun 18. Bioorg Med Chem Lett. 2019. PMID: 31272790
Bridelia speciosa Müll.Arg. Stem bark Extracts as a Potential Biomedicine: From Tropical Western Africa to the Pharmacy Shelf.
Mahomoodally MF, Sinan KI, Bene K, Zengin G, Orlando G, Menghini L, Veschi S, Chiavaroli A, Recinella L, Brunetti L, Leone S, Angelini P, Hubka V, Covino S, Venanzoni R, Picot-Allain MCN, Lellis L, Cama A, Cziáky Z, Jekő J, Ferrante C. Mahomoodally MF, et al. Among authors: cama a. Antioxidants (Basel). 2020 Feb 2;9(2):128. doi: 10.3390/antiox9020128. Antioxidants (Basel). 2020. PMID: 32024319 Free PMC article.
Sulfonimide and Amide Derivatives as Novel PPARα Antagonists: Synthesis, Antiproliferative Activity, and Docking Studies.
Ammazzalorso A, Bruno I, Florio R, De Lellis L, Laghezza A, Cerchia C, De Filippis B, Fantacuzzi M, Giampietro L, Maccallini C, Tortorella P, Veschi S, Loiodice F, Lavecchia A, Cama A, Amoroso R. Ammazzalorso A, et al. Among authors: cama a. ACS Med Chem Lett. 2020 Mar 3;11(5):624-632. doi: 10.1021/acsmedchemlett.9b00666. eCollection 2020 May 14. ACS Med Chem Lett. 2020. PMID: 32435362 Free PMC article.
Protective Effects Induced by a Hydroalcoholic Allium sativum Extract in Isolated Mouse Heart.
Recinella L, Chiavaroli A, Masciulli F, Fraschetti C, Filippi A, Cesa S, Cairone F, Gorica E, De Leo M, Braca A, Martelli A, Calderone V, Orlando G, Ferrante C, Menghini L, Di Simone SC, Veschi S, Cama A, Brunetti L, Leone S. Recinella L, et al. Among authors: cama a. Nutrients. 2021 Jul 8;13(7):2332. doi: 10.3390/nu13072332. Nutrients. 2021. PMID: 34371842 Free PMC article.
Benzothiazole Derivatives Endowed with Antiproliferative Activity in Paraganglioma and Pancreatic Cancer Cells: Structure-Activity Relationship Studies and Target Prediction Analysis.
Amoroso R, De Lellis L, Florio R, Moreno N, Agamennone M, De Filippis B, Giampietro L, Maccallini C, Fernández I, Recio R, Cama A, Fantacuzzi M, Ammazzalorso A. Amoroso R, et al. Among authors: cama a. Pharmaceuticals (Basel). 2022 Jul 28;15(8):937. doi: 10.3390/ph15080937. Pharmaceuticals (Basel). 2022. PMID: 36015085 Free PMC article.
A grape (Vitis vinifera L.) pomace water extract modulates inflammatory and immune response in SW-480 cells and isolated mouse colon.
Recinella L, Chiavaroli A, Veschi S, Cama A, Acquaviva A, Libero ML, Leone S, Di Simone SC, Pagano E, Zengin G, Menghini L, Brunetti L, Izzo AA, Orlando G, Ferrante C. Recinella L, et al. Among authors: cama a. Phytother Res. 2022 Dec;36(12):4620-4630. doi: 10.1002/ptr.7581. Epub 2022 Sep 7. Phytother Res. 2022. PMID: 36069605 Free PMC article.
Synthesis, in vitro evaluation, and molecular modeling investigation of benzenesulfonimide peroxisome proliferator-activated receptors α antagonists.
Ammazzalorso A, Carrieri A, Verginelli F, Bruno I, Carbonara G, D'Angelo A, De Filippis B, Fantacuzzi M, Florio R, Fracchiolla G, Giampietro L, Giancristofaro A, Maccallini C, Cama A, Amoroso R. Ammazzalorso A, et al. Among authors: cama a. Eur J Med Chem. 2016 May 23;114:191-200. doi: 10.1016/j.ejmech.2016.02.064. Epub 2016 Feb 27. Eur J Med Chem. 2016. PMID: 26974385
359 results