Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
7 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Multitargeting application of proline-derived peptidomimetics addressing cancer-related human matrix metalloproteinase 9 and carbonic anhydrase II.
Eur J Med Chem. 2021 Mar 15;214:113260. doi: 10.1016/j.ejmech.2021.113260. Epub 2021 Feb 4.
Eur J Med Chem. 2021.
PMID: 33581552
Synthesis of morpholine derivatives using the Castagnoli-Cushman reaction as BACE1 inhibitors: Unexpected binding activity of cyclic thioamides.
Calugi L, Lenci E, Innocenti R, Trabocchi A.
Calugi L, et al.
Bioorg Med Chem Lett. 2020 Jul 1;30(13):127211. doi: 10.1016/j.bmcl.2020.127211. Epub 2020 Apr 24.
Bioorg Med Chem Lett. 2020.
PMID: 32354570
Item in Clipboard
Computational-aided design of a library of lactams through a diversity-oriented synthesis strategy.
Saldívar-González FI, Lenci E, Calugi L, Medina-Franco JL, Trabocchi A.
Saldívar-González FI, et al. Among authors: calugi l.
Bioorg Med Chem. 2020 Jun 15;28(12):115539. doi: 10.1016/j.bmc.2020.115539. Epub 2020 May 4.
Bioorg Med Chem. 2020.
PMID: 32503698
Item in Clipboard
Occurrence of Morpholine in Central Nervous System Drug Discovery.
Lenci E, Calugi L, Trabocchi A.
Lenci E, et al. Among authors: calugi l.
ACS Chem Neurosci. 2021 Feb 3;12(3):378-390. doi: 10.1021/acschemneuro.0c00729. Epub 2021 Jan 18.
ACS Chem Neurosci. 2021.
PMID: 33459557
Free PMC article.
Item in Clipboard
Peptidomimetic Small-Molecule Inhibitors of 3CLPro Activity and Spike-ACE2 Interaction: Toward Dual-Action Molecules against Coronavirus Infections.
Tedesco F, Calugi L, Lenci E, Trabocchi A.
Tedesco F, et al. Among authors: calugi l.
J Org Chem. 2022 Sep 16;87(18):12041-12051. doi: 10.1021/acs.joc.2c01047. Epub 2022 Aug 30.
J Org Chem. 2022.
PMID: 36039955
Free PMC article.
Item in Clipboard
Modular synthesis of 2,4-diaminoanilines as CNS drug-like non-covalent inhibitors of asparagine endopeptidase.
Calugi L, Lenci E, Bianchini F, Contini A, Trabocchi A.
Calugi L, et al.
Bioorg Med Chem. 2022 Jun 1;63:116746. doi: 10.1016/j.bmc.2022.116746. Epub 2022 Apr 12.
Bioorg Med Chem. 2022.
PMID: 35430537
Item in Clipboard
Identification of a short ACE2-derived stapled peptide targeting the SARS-CoV-2 spike protein.
Calugi L, Sautariello G, Lenci E, Mattei ML, Coppa C, Cini N, Contini A, Trabocchi A.
Calugi L, et al.
Eur J Med Chem. 2023 Mar 5;249:115118. doi: 10.1016/j.ejmech.2023.115118. Epub 2023 Jan 17.
Eur J Med Chem. 2023.
PMID: 36682293
Free PMC article.
Item in Clipboard
Cite
Cite