Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
6 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Synthesis and biological evaluation of analogues of 7-chloro-4,5-dihydro-4- oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylic acid (TQX-173) as novel selective AMPA receptor antagonists.
J Med Chem. 2004 Jan 1;47(1):262-72. doi: 10.1021/jm030906q.
J Med Chem. 2004.
PMID: 14695840
3-hydroxy-quinazoline-2,4-dione as a useful scaffold to obtain selective Gly/NMDA and AMPA receptor antagonists.
Colotta V, Catarzi D, Varano F, Calabri FR, Filacchioni G, Costagli C, Galli A.
Colotta V, et al. Among authors: calabri fr.
Bioorg Med Chem Lett. 2004 May 3;14(9):2345-9. doi: 10.1016/j.bmcl.2004.01.109.
Bioorg Med Chem Lett. 2004.
PMID: 15081038
Item in Clipboard
1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies.
Colotta V, Catarzi D, Varano F, Calabri FR, Lenzi O, Filacchioni G, Martini C, Trincavelli L, Deflorian F, Moro S.
Colotta V, et al. Among authors: calabri fr.
J Med Chem. 2004 Jul 1;47(14):3580-90. doi: 10.1021/jm031136l.
J Med Chem. 2004.
PMID: 15214785
Item in Clipboard
2-aryl-8-chloro-1,2,4-triazolo[1,5-a]quinoxalin-4-amines as highly potent A1 and A3 adenosine receptor antagonists.
Catarzi D, Colotta V, Varano F, Calabri FR, Lenzi O, Filacchioni G, Trincavelli L, Martini C, Tralli A, Montopoli C, Moro S.
Catarzi D, et al. Among authors: calabri fr.
Bioorg Med Chem. 2005 Feb 1;13(3):705-15. doi: 10.1016/j.bmc.2004.10.050.
Bioorg Med Chem. 2005.
PMID: 15653338
Item in Clipboard
Synthesis and pharmacological studies at the Gly/NMDA, AMPA and Kainate receptors of new oxazolo[4,5-c]quinolin-4-one derivatives bearing different substituents at position-2 and on the fused benzo ring.
Calabri FR, Colotta V, Catarzi D, Varano F, Lenzi O, Filacchioni G, Costagli C, Galli A.
Calabri FR, et al.
Eur J Med Chem. 2005 Sep;40(9):897-907. doi: 10.1016/j.ejmech.2005.03.017.
Eur J Med Chem. 2005.
PMID: 15919134
Item in Clipboard
1-Substituted pyrazolo[1,5-c]quinazolines as novel Gly/NMDA receptor antagonists: synthesis, biological evaluation, and molecular modeling study.
Varano F, Catarzi D, Colotta V, Calabri FR, Lenzi O, Filacchioni G, Galli A, Costagli C, Deflorian F, Moro S.
Varano F, et al. Among authors: calabri fr.
Bioorg Med Chem. 2005 Oct 1;13(19):5536-49. doi: 10.1016/j.bmc.2005.07.010.
Bioorg Med Chem. 2005.
PMID: 16087341
Item in Clipboard
Cite
Cite