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Targeting BER enzymes in cancer therapy.
DNA Repair (Amst). 2018 Nov;71:118-126. doi: 10.1016/j.dnarep.2018.08.015. Epub 2018 Aug 25.
DNA Repair (Amst). 2018.
PMID: 30228084
Free article.
Review.
Targeting OGG1 arrests cancer cell proliferation by inducing replication stress.
Visnes T, Benítez-Buelga C, Cázares-Körner A, Sanjiv K, Hanna BMF, Mortusewicz O, Rajagopal V, Albers JJ, Hagey DW, Bekkhus T, Eshtad S, Baquero JM, Masuyer G, Wallner O, Müller S, Pham T, Göktürk C, Rasti A, Suman S, Torres-Ruiz R, Sarno A, Wiita E, Homan EJ, Karsten S, Marimuthu K, Michel M, Koolmeister T, Scobie M, Loseva O, Almlöf I, Unterlass JE, Pettke A, Boström J, Pandey M, Gad H, Herr P, Jemth AS, El Andaloussi S, Kalderén C, Rodriguez-Perales S, Benítez J, Krokan HE, Altun M, Stenmark P, Berglund UW, Helleday T.
Visnes T, et al. Among authors: cazares korner a.
Nucleic Acids Res. 2020 Dec 2;48(21):12234-12251. doi: 10.1093/nar/gkaa1048.
Nucleic Acids Res. 2020.
PMID: 33211885
Free PMC article.
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Small-molecule inhibitor of OGG1 suppresses proinflammatory gene expression and inflammation.
Visnes T, Cázares-Körner A, Hao W, Wallner O, Masuyer G, Loseva O, Mortusewicz O, Wiita E, Sarno A, Manoilov A, Astorga-Wells J, Jemth AS, Pan L, Sanjiv K, Karsten S, Gokturk C, Grube M, Homan EJ, Hanna BMF, Paulin CBJ, Pham T, Rasti A, Berglund UW, von Nicolai C, Benitez-Buelga C, Koolmeister T, Ivanic D, Iliev P, Scobie M, Krokan HE, Baranczewski P, Artursson P, Altun M, Jensen AJ, Kalderén C, Ba X, Zubarev RA, Stenmark P, Boldogh I, Helleday T.
Visnes T, et al. Among authors: cazares korner a.
Science. 2018 Nov 16;362(6416):834-839. doi: 10.1126/science.aar8048.
Science. 2018.
PMID: 30442810
Free PMC article.
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Novel Broad-Spectrum Antiviral Inhibitors Targeting Host Factors Essential for Replication of Pathogenic RNA Viruses.
Tampere M, Pettke A, Salata C, Wallner O, Koolmeister T, Cazares-Körner A, Visnes T, Hesselman MC, Kunold E, Wiita E, Kalderén C, Lightowler M, Jemth AS, Lehtiö J, Rosenquist Å, Warpman-Berglund U, Helleday T, Mirazimi A, Jafari R, Puumalainen MR.
Tampere M, et al. Among authors: cazares korner a.
Viruses. 2020 Dec 10;12(12):1423. doi: 10.3390/v12121423.
Viruses. 2020.
PMID: 33322045
Free PMC article.
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Optimization of N-Piperidinyl-Benzimidazolone Derivatives as Potent and Selective Inhibitors of 8-Oxo-Guanine DNA Glycosylase 1.
Wallner O, Cázares-Körner A, Scaletti ER, Masuyer G, Bekkhus T, Visnes T, Mamonov K, Ortis F, Lundbäck T, Volkova M, Koolmeister T, Wiita E, Loseva O, Pandey M, Homan E, Benítez-Buelga C, Davies J, Scobie M, Warpman Berglund U, Kalderén C, Stenmark P, Helleday T, Michel M.
Wallner O, et al. Among authors: cazares korner a.
ChemMedChem. 2023 Jan 3;18(1):e202200310. doi: 10.1002/cmdc.202200310. Epub 2022 Oct 13.
ChemMedChem. 2023.
PMID: 36128847
Free PMC article.
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Development of a chemical probe against NUDT15.
Zhang SM, Desroses M, Hagenkort A, Valerie NCK, Rehling D, Carter M, Wallner O, Koolmeister T, Throup A, Jemth AS, Almlöf I, Loseva O, Lundbäck T, Axelsson H, Regmi S, Sarno A, Krämer A, Pudelko L, Bräutigam L, Rasti A, Göttmann M, Wiita E, Kutzner J, Schaller T, Kalderén C, Cázares-Körner A, Page BDG, Krimpenfort R, Eshtad S, Altun M, Rudd SG, Knapp S, Scobie M, Homan EJ, Berglund UW, Stenmark P, Helleday T.
Zhang SM, et al. Among authors: cazares korner a.
Nat Chem Biol. 2020 Oct;16(10):1120-1128. doi: 10.1038/s41589-020-0592-z. Epub 2020 Jul 20.
Nat Chem Biol. 2020.
PMID: 32690945
Free PMC article.
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Engineering transketolase to accept both unnatural donor and acceptor substrates and produce α-hydroxyketones.
Yu H, Hernández López RI, Steadman D, Méndez-Sánchez D, Higson S, Cázares-Körner A, Sheppard TD, Ward JM, Hailes HC, Dalby PA.
Yu H, et al. Among authors: cazares korner a.
FEBS J. 2020 May;287(9):1758-1776. doi: 10.1111/febs.15108. Epub 2019 Nov 10.
FEBS J. 2020.
PMID: 31647171
Free article.
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Multi-step biocatalytic strategies for chiral amino alcohol synthesis.
Villegas-Torres MF, Martinez-Torres RJ, Cázares-Körner A, Hailes H, Baganz F, Ward J.
Villegas-Torres MF, et al. Among authors: cazares korner a.
Enzyme Microb Technol. 2015 Dec;81:23-30. doi: 10.1016/j.enzmictec.2015.07.003. Epub 2015 Jul 10.
Enzyme Microb Technol. 2015.
PMID: 26453469
Free article.
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