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Grafting aminocyclopentane carboxylic acids onto the RGD tripeptide sequence generates low nanomolar alphaVbeta3/alphaVbeta5 integrin dual binders.
J Med Chem. 2005 Dec 1;48(24):7675-87. doi: 10.1021/jm050698x.
J Med Chem. 2005.
PMID: 16302808
Targeting alphavbeta3 integrin: design and applications of mono- and multifunctional RGD-based peptides and semipeptides.
Auzzas L, Zanardi F, Battistini L, Burreddu P, Carta P, Rassu G, Curti C, Casiraghi G.
Auzzas L, et al. Among authors: burreddu p.
Curr Med Chem. 2010;17(13):1255-99. doi: 10.2174/092986710790936301.
Curr Med Chem. 2010.
PMID: 20166941
Review.
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Discovery of subnanomolar arginine-glycine-aspartate-based alphaVbeta3/alphaVbeta5 integrin binders embedding 4-aminoproline residues.
Zanardi F, Burreddu P, Rassu G, Auzzas L, Battistini L, Curti C, Sartori A, Nicastro G, Menchi G, Cini N, Bottoncetti A, Raspanti S, Casiraghi G.
Zanardi F, et al. Among authors: burreddu p.
J Med Chem. 2008 Mar 27;51(6):1771-82. doi: 10.1021/jm701214z. Epub 2008 Feb 28.
J Med Chem. 2008.
PMID: 18303826
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4-Aminoproline-based arginine-glycine-aspartate integrin binders with exposed ligation points: practical in-solution synthesis, conjugation and binding affinity evaluation.
Battistini L, Burreddu P, Carta P, Rassu G, Auzzas L, Curti C, Zanardi F, Manzoni L, Araldi EM, Scolastico C, Casiraghi G.
Battistini L, et al. Among authors: burreddu p.
Org Biomol Chem. 2009 Dec 7;7(23):4924-35. doi: 10.1039/b914836a. Epub 2009 Oct 6.
Org Biomol Chem. 2009.
PMID: 19907783
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Variable strategy toward carbasugars and relatives. 6. Diastereoselective synthesis of 2-deoxy-2-amino-5a-carba-beta-L-mannopyranuronic acid and 2-deoxy-2-amino-5a-carba-beta-L-mannopyranose.
Rassu G, Auzzas L, Zambrano V, Burreddu P, Pinna L, Battistini L, Zanardi F, Casiraghi G.
Rassu G, et al. Among authors: burreddu p.
J Org Chem. 2004 Mar 5;69(5):1625-8. doi: 10.1021/jo0357216.
J Org Chem. 2004.
PMID: 14987021
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Vicarious silylative Mukaiyama aldol reaction: a vinylogous extension.
Curti C, Sartori A, Battistini L, Rassu G, Burreddu P, Zanardi F, Casiraghi G.
Curti C, et al. Among authors: burreddu p.
J Org Chem. 2008 Jul 18;73(14):5446-51. doi: 10.1021/jo800741c. Epub 2008 Jun 13.
J Org Chem. 2008.
PMID: 18549289
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Design, synthesis, and biological evaluation of novel cRGD-paclitaxel conjugates for integrin-assisted drug delivery.
Pilkington-Miksa M, Arosio D, Battistini L, Belvisi L, De Matteo M, Vasile F, Burreddu P, Carta P, Rassu G, Perego P, Carenini N, Zunino F, De Cesare M, Castiglioni V, Scanziani E, Scolastico C, Casiraghi G, Zanardi F, Manzoni L.
Pilkington-Miksa M, et al. Among authors: burreddu p.
Bioconjug Chem. 2012 Aug 15;23(8):1610-22. doi: 10.1021/bc300164t. Epub 2012 Jul 20.
Bioconjug Chem. 2012.
PMID: 22770429
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Enhancement of the uptake and cytotoxic activity of doxorubicin in cancer cells by novel cRGD-semipeptide-anchoring liposomes.
Battistini L, Burreddu P, Sartori A, Arosio D, Manzoni L, Paduano L, D'Errico G, Sala R, Reia L, Bonomini S, Rassu G, Zanardi F.
Battistini L, et al. Among authors: burreddu p.
Mol Pharm. 2014 Jul 7;11(7):2280-93. doi: 10.1021/mp400718j. Epub 2014 May 22.
Mol Pharm. 2014.
PMID: 24819754
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