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Antitumor activity of bis-indole derivatives.
Andreani A, Burnelli S, Granaiola M, Leoni A, Locatelli A, Morigi R, Rambaldi M, Varoli L, Landi L, Prata C, Berridge MV, Grasso C, Fiebig HH, Kelter G, Burger AM, Kunkel MW. Andreani A, et al. Among authors: burnelli s. J Med Chem. 2008 Aug 14;51(15):4563-70. doi: 10.1021/jm800194k. Epub 2008 Jul 4. J Med Chem. 2008. PMID: 18598018 Free PMC article.
Chemiluminescent high-throughput microassay applied to imidazo[2,1-b]thiazole derivatives as potential acetylcholinesterase and butyrylcholinesterase inhibitors.
Andreani A, Burnelli S, Granaiola M, Guardigli M, Leoni A, Locatelli A, Morigi R, Rambaldi M, Rizzoli M, Varoli L, Roda A. Andreani A, et al. Among authors: burnelli s. Eur J Med Chem. 2008 Mar;43(3):657-61. doi: 10.1016/j.ejmech.2007.04.018. Epub 2007 May 21. Eur J Med Chem. 2008. PMID: 17624631
New antitumor imidazo[2,1-b]thiazole guanylhydrazones and analogues.
Andreani A, Burnelli S, Granaiola M, Leoni A, Locatelli A, Morigi R, Rambaldi M, Varoli L, Calonghi N, Cappadone C, Farruggia G, Zini M, Stefanelli C, Masotti L, Radin NS, Shoemaker RH. Andreani A, et al. Among authors: burnelli s. J Med Chem. 2008 Feb 28;51(4):809-16. doi: 10.1021/jm701246g. Epub 2008 Feb 6. J Med Chem. 2008. PMID: 18251494
Diphenidol-related diamines as novel muscarinic M4 receptor antagonists.
Varoli L, Andreani A, Burnelli S, Granaiola M, Leoni A, Locatelli A, Morigi R, Rambaldi M, Bedini A, Fazio N, Spampinato S. Varoli L, et al. Among authors: burnelli s. Bioorg Med Chem Lett. 2008 May 1;18(9):2972-6. doi: 10.1016/j.bmcl.2008.03.061. Epub 2008 Mar 23. Bioorg Med Chem Lett. 2008. PMID: 18395442
Antitumor activity of new substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones and 3-(5-imidazo[2,1-b]thiadiazolylmethylene)-2-indolinones: selectivity against colon tumor cells and effect on cell cycle-related events.
Andreani A, Burnelli S, Granaiola M, Leoni A, Locatelli A, Morigi R, Rambaldi M, Varoli L, Calonghi N, Cappadone C, Voltattorni M, Zini M, Stefanelli C, Masotti L, Shoemaker RH. Andreani A, et al. Among authors: burnelli s. J Med Chem. 2008 Dec 11;51(23):7508-13. doi: 10.1021/jm800827q. J Med Chem. 2008. PMID: 19006285
New isatin derivatives with antioxidant activity.
Andreani A, Burnelli S, Granaiola M, Leoni A, Locatelli A, Morigi R, Rambaldi M, Varoli L, Cremonini MA, Placucci G, Cervellati R, Greco E. Andreani A, et al. Among authors: burnelli s. Eur J Med Chem. 2010 Apr;45(4):1374-8. doi: 10.1016/j.ejmech.2009.12.035. Epub 2009 Dec 28. Eur J Med Chem. 2010. PMID: 20060202
Antitumor activity and COMPARE analysis of bis-indole derivatives.
Andreani A, Burnelli S, Granaiola M, Leoni A, Locatelli A, Morigi R, Rambaldi M, Varoli L, Landi L, Prata C, Dalla Sega FV, Caliceti C, Shoemaker RH. Andreani A, et al. Among authors: burnelli s. Bioorg Med Chem. 2010 May 1;18(9):3004-11. doi: 10.1016/j.bmc.2010.03.063. Epub 2010 Mar 28. Bioorg Med Chem. 2010. PMID: 20395150
39 results