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Impaired expression of serine/arginine protein kinase 2 (SRPK2) affects melanoma progression.
Caetano MMM, Moreira GA, da Silva MR, Guimarães GR, Santos LO, Pacheco AA, Siqueira RP, Mendes FC, Marques Da Silva EA, Junior AS, Rangel Fietto JL, Saito Â, Boroni M, Bressan GC. Caetano MMM, et al. Among authors: bressan gc. Front Genet. 2022 Sep 23;13:979735. doi: 10.3389/fgene.2022.979735. eCollection 2022. Front Genet. 2022. PMID: 36212152 Free PMC article.
Potential Antileukemia Effect and Structural Analyses of SRPK Inhibition by N-(2-(Piperidin-1-yl)-5-(Trifluoromethyl)Phenyl)Isonicotinamide (SRPIN340).
Siqueira RP, Barbosa Éde A, Polêto MD, Righetto GL, Seraphim TV, Salgado RL, Ferreira JG, Barros MV, de Oliveira LL, Laranjeira AB, Almeida MR, Júnior AS, Fietto JL, Kobarg J, de Oliveira EB, Teixeira RR, Borges JC, Yunes JA, Bressan GC. Siqueira RP, et al. Among authors: bressan gc. PLoS One. 2015 Aug 5;10(8):e0134882. doi: 10.1371/journal.pone.0134882. eCollection 2015. PLoS One. 2015. PMID: 26244849 Free PMC article.
Splicing Regulators and Their Roles in Cancer Biology and Therapy.
da Silva MR, Moreira GA, Gonçalves da Silva RA, de Almeida Alves Barbosa É, Pais Siqueira R, Teixera RR, Almeida MR, Silva Júnior A, Fietto JL, Bressan GC. da Silva MR, et al. Among authors: bressan gc. Biomed Res Int. 2015;2015:150514. doi: 10.1155/2015/150514. Epub 2015 Jul 26. Biomed Res Int. 2015. PMID: 26273588 Free PMC article. Review.
Synthesis, molecular properties prediction and cytotoxic screening of 3-(2-aryl-2-oxoethyl)isobenzofuran-1(3H)-ones.
da Silva Maia AF, Siqueira RP, de Oliveira FM, Ferreira JG, da Silva SF, Caiuby CAD, de Oliveira LL, de Paula SO, Souza RAC, Guilardi S, Bressan GC, Teixeira RR. da Silva Maia AF, et al. Among authors: bressan gc. Bioorg Med Chem Lett. 2016 Jun 15;26(12):2810-2816. doi: 10.1016/j.bmcl.2016.04.065. Epub 2016 Apr 25. Bioorg Med Chem Lett. 2016. PMID: 27155902
Trifluoromethyl arylamides with antileukemia effect and intracellular inhibitory activity over serine/arginine-rich protein kinases (SRPKs).
Siqueira RP, Barros MVA, Barbosa ÉAA, Onofre TS, Gonçalves VHS, Pereira HS, Silva Júnior A, de Oliveira LL, Almeida MR, Fietto JLR, Teixeira RR, Bressan GC. Siqueira RP, et al. Among authors: bressan gc. Eur J Med Chem. 2017 Jul 7;134:97-109. doi: 10.1016/j.ejmech.2017.03.078. Epub 2017 Mar 31. Eur J Med Chem. 2017. PMID: 28407594
84 results