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Leishmanicidal and cytotoxic activities and 4D-QSAR of 2-arylidene indan-1,3-diones.
de Souza APM, Costa MCA, de Aguiar AR, Bressan GC, de Almeida Lima GD, Lima WP, Borsodi MPG, Bergmann BR, Ferreira MMC, Teixeira RR. de Souza APM, et al. Among authors: bressan gc. Arch Pharm (Weinheim). 2021 Oct;354(10):e2100081. doi: 10.1002/ardp.202100081. Epub 2021 Jul 29. Arch Pharm (Weinheim). 2021. PMID: 34323311
Potential Antileukemia Effect and Structural Analyses of SRPK Inhibition by N-(2-(Piperidin-1-yl)-5-(Trifluoromethyl)Phenyl)Isonicotinamide (SRPIN340).
Siqueira RP, Barbosa Éde A, Polêto MD, Righetto GL, Seraphim TV, Salgado RL, Ferreira JG, Barros MV, de Oliveira LL, Laranjeira AB, Almeida MR, Júnior AS, Fietto JL, Kobarg J, de Oliveira EB, Teixeira RR, Borges JC, Yunes JA, Bressan GC. Siqueira RP, et al. Among authors: bressan gc. PLoS One. 2015 Aug 5;10(8):e0134882. doi: 10.1371/journal.pone.0134882. eCollection 2015. PLoS One. 2015. PMID: 26244849 Free PMC article.
The Antileishmanial Potential of C-3 Functionalized Isobenzofuranones against Leishmania (Leishmania) Infantum Chagasi.
Pereira WL, de Souza Vasconcellos R, Mariotini-Moura C, Saar Gomes R, Firmino Rde C, da Silva AM, Silva Júnior A, Bressan GC, Almeida MR, Crocco Afonso LC, Teixeira RR, Lopes Rangel Fietto J. Pereira WL, et al. Among authors: bressan gc. Molecules. 2015 Dec 14;20(12):22435-44. doi: 10.3390/molecules201219857. Molecules. 2015. PMID: 26694330 Free PMC article.
Synthesis, molecular properties prediction and cytotoxic screening of 3-(2-aryl-2-oxoethyl)isobenzofuran-1(3H)-ones.
da Silva Maia AF, Siqueira RP, de Oliveira FM, Ferreira JG, da Silva SF, Caiuby CAD, de Oliveira LL, de Paula SO, Souza RAC, Guilardi S, Bressan GC, Teixeira RR. da Silva Maia AF, et al. Among authors: bressan gc. Bioorg Med Chem Lett. 2016 Jun 15;26(12):2810-2816. doi: 10.1016/j.bmcl.2016.04.065. Epub 2016 Apr 25. Bioorg Med Chem Lett. 2016. PMID: 27155902
Trifluoromethyl arylamides with antileukemia effect and intracellular inhibitory activity over serine/arginine-rich protein kinases (SRPKs).
Siqueira RP, Barros MVA, Barbosa ÉAA, Onofre TS, Gonçalves VHS, Pereira HS, Silva Júnior A, de Oliveira LL, Almeida MR, Fietto JLR, Teixeira RR, Bressan GC. Siqueira RP, et al. Among authors: bressan gc. Eur J Med Chem. 2017 Jul 7;134:97-109. doi: 10.1016/j.ejmech.2017.03.078. Epub 2017 Mar 31. Eur J Med Chem. 2017. PMID: 28407594
Antimetastatic effect of the pharmacological inhibition of serine/arginine-rich protein kinases (SRPK) in murine melanoma.
Moreira GA, Lima GDA, Siqueira RP, Barros MVA, Adjanohoun ALM, Santos VC, Barbosa ÉAA, Loterio RK, Paiva JC, Gonçalves VHS, Viol LCS, Marques-da-Silva EA, Júnior AS, Almeida MR, Fietto JLR, Machado-Neves M, Ferreira RS, Teixeira RR, Bressan GC. Moreira GA, et al. Among authors: bressan gc. Toxicol Appl Pharmacol. 2018 Oct 1;356:214-223. doi: 10.1016/j.taap.2018.08.012. Epub 2018 Aug 20. Toxicol Appl Pharmacol. 2018. PMID: 30138656 Free article.
Synthesis of cinnamic acid derivatives and leishmanicidal activity against Leishmania braziliensis.
Rodrigues MP, Tomaz DC, Ângelo de Souza L, Onofre TS, Aquiles de Menezes W, Almeida-Silva J, Suarez-Fontes AM, Rogéria de Almeida M, Manoel da Silva A, Bressan GC, Vannier-Santos MA, Rangel Fietto JL, Teixeira RR. Rodrigues MP, et al. Among authors: bressan gc. Eur J Med Chem. 2019 Dec 1;183:111688. doi: 10.1016/j.ejmech.2019.111688. Epub 2019 Sep 9. Eur J Med Chem. 2019. PMID: 31542714
84 results