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Glycine-replaced derivatives of [Pro3,DLeu9]TL, a temporin L analogue: Evaluation of antimicrobial, cytotoxic and hemolytic activities.
Merlino F, Carotenuto A, Casciaro B, Martora F, Loffredo MR, Di Grazia A, Yousif AM, Brancaccio D, Palomba L, Novellino E, Galdiero M, Iovene MR, Mangoni ML, Grieco P. Merlino F, et al. Among authors: brancaccio d. Eur J Med Chem. 2017 Oct 20;139:750-761. doi: 10.1016/j.ejmech.2017.08.040. Epub 2017 Aug 21. Eur J Med Chem. 2017. PMID: 28863356
New insight into the binding mode of peptide ligands at Urotensin-II receptor: structure-activity relationships study on P5U and urantide.
Grieco P, Carotenuto A, Campiglia P, Gomez-Monterrey I, Auriemma L, Sala M, Marcozzi C, d'Emmanuele di Villa Bianca R, Brancaccio D, Rovero P, Santicioli P, Meini S, Maggi CA, Novellino E. Grieco P, et al. Among authors: d emmanuele di villa bianca r, brancaccio d. J Med Chem. 2009 Jul 9;52(13):3927-40. doi: 10.1021/jm900148c. J Med Chem. 2009. PMID: 19432421
Design, synthesis, and cytotoxic evaluation of acyl derivatives of 3-aminonaphtho[2,3-b]thiophene-4,9-dione, a quinone-based system.
Gomez-Monterrey I, Campiglia P, Aquino C, Bertamino A, Granata I, Carotenuto A, Brancaccio D, Stiuso P, Scognamiglio I, Rusciano MR, Maione AS, Illario M, Grieco P, Maresca B, Novellino E. Gomez-Monterrey I, et al. Among authors: brancaccio d. J Med Chem. 2011 Jun 23;54(12):4077-91. doi: 10.1021/jm200094h. Epub 2011 May 23. J Med Chem. 2011. PMID: 21553829
Development of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors.
Merlino F, Zhou Y, Cai M, Carotenuto A, Yousif AM, Brancaccio D, Di Maro S, Zappavigna S, Limatola A, Novellino E, Grieco P, Hruby VJ. Merlino F, et al. Among authors: brancaccio d. J Med Chem. 2018 May 10;61(9):4263-4269. doi: 10.1021/acs.jmedchem.8b00488. Epub 2018 Apr 25. J Med Chem. 2018. PMID: 29660981 Free PMC article.
The Outcomes of Decorated Prolines in the Discovery of Antimicrobial Peptides from Temporin-L.
Buommino E, Carotenuto A, Antignano I, Bellavita R, Casciaro B, Loffredo MR, Merlino F, Novellino E, Mangoni ML, Nocera FP, Brancaccio D, Punzi P, Roversi D, Ingenito R, Bianchi E, Grieco P. Buommino E, et al. Among authors: brancaccio d. ChemMedChem. 2019 Jul 3;14(13):1283-1290. doi: 10.1002/cmdc.201900221. Epub 2019 Jun 3. ChemMedChem. 2019. PMID: 31087626
First-in-Class Cyclic Temporin L Analogue: Design, Synthesis, and Antimicrobial Assessment.
Bellavita R, Casciaro B, Di Maro S, Brancaccio D, Carotenuto A, Falanga A, Cappiello F, Buommino E, Galdiero S, Novellino E, Grossmann TN, Mangoni ML, Merlino F, Grieco P. Bellavita R, et al. Among authors: brancaccio d. J Med Chem. 2021 Aug 12;64(15):11675-11694. doi: 10.1021/acs.jmedchem.1c01033. Epub 2021 Jul 23. J Med Chem. 2021. PMID: 34296619 Free PMC article.
Identification of the spiro(oxindole-3,3'-thiazolidine)-based derivatives as potential p53 activity modulators.
Gomez-Monterrey I, Bertamino A, Porta A, Carotenuto A, Musella S, Aquino C, Granata I, Sala M, Brancaccio D, Picone D, Ercole C, Stiuso P, Campiglia P, Grieco P, Ianelli P, Maresca B, Novellino E. Gomez-Monterrey I, et al. Among authors: brancaccio d. J Med Chem. 2010 Dec 9;53(23):8319-29. doi: 10.1021/jm100838z. Epub 2010 Nov 8. J Med Chem. 2010. PMID: 21058726
279 results