Braconi L - Search Results

1

Application of LEDA algorithm for the recognition of P-glycoprotein and Carbonic Anhydrase hybrid inhibitors and evaluation of their plasma stability by HPLC-MS/MS analysis.

Pallecchi M, Menicatti M, Braconi L, Supuran CT, Dei S, Teodori E, Bartolucci G. Pallecchi M, et al. Among authors: braconi l. J Pharm Biomed Anal. 2022 Sep 20;219:114887. doi: 10.1016/j.jpba.2022.114887. Epub 2022 Jun 10. J Pharm Biomed Anal. 2022. PMID: 35753165

2

Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug resistance (MDR) modulators.

Dei S, Braconi L, Trezza A, Menicatti M, Contino M, Coronnello M, Chiaramonte N, Manetti D, Perrone MG, Romanelli MN, Udomtanakunchai C, Colabufo NA, Bartolucci G, Spiga O, Salerno M, Teodori E. Dei S, et al. Among authors: braconi l. Eur J Med Chem. 2019 Jun 15;172:71-94. doi: 10.1016/j.ejmech.2019.03.054. Epub 2019 Mar 27. Eur J Med Chem. 2019. PMID: 30947123

3

Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors.

Chiaramonte N, Bua S, Angeli A, Ferraroni M, Picchioni I, Bartolucci G, Braconi L, Dei S, Teodori E, Supuran CT, Romanelli MN. Chiaramonte N, et al. Among authors: braconi l. Bioorg Chem. 2019 Oct;91:103130. doi: 10.1016/j.bioorg.2019.103130. Epub 2019 Jul 20. Bioorg Chem. 2019. PMID: 31374520

4

Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers.

Teodori E, Contino M, Riganti C, Bartolucci G, Braconi L, Manetti D, Romanelli MN, Trezza A, Athanasios A, Spiga O, Perrone MG, Giampietro R, Gazzano E, Salerno M, Colabufo NA, Dei S. Teodori E, et al. Among authors: braconi l. Eur J Med Chem. 2019 Nov 15;182:111655. doi: 10.1016/j.ejmech.2019.111655. Epub 2019 Aug 30. Eur J Med Chem. 2019. PMID: 31494468

5

6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers.

Braconi L, Bartolucci G, Contino M, Chiaramonte N, Giampietro R, Manetti D, Perrone MG, Romanelli MN, Colabufo NA, Riganti C, Dei S, Teodori E. Braconi L, et al. J Enzyme Inhib Med Chem. 2020 Dec;35(1):974-992. doi: 10.1080/14756366.2020.1747449. J Enzyme Inhib Med Chem. 2020. PMID: 32253945 Free PMC article.

6

Dual P-Glycoprotein and CA XII Inhibitors: A New Strategy to Reverse the P-gp Mediated Multidrug Resistance (MDR) in Cancer Cells.

Teodori E, Braconi L, Bua S, Lapucci A, Bartolucci G, Manetti D, Romanelli MN, Dei S, Supuran CT, Coronnello M. Teodori E, et al. Among authors: braconi l. Molecules. 2020 Apr 10;25(7):1748. doi: 10.3390/molecules25071748. Molecules. 2020. PMID: 32290281 Free PMC article.

7

Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine¹.

Chiaramonte N, Maach S, Biliotti C, Angeli A, Bartolucci G, Braconi L, Dei S, Teodori E, Supuran CT, Romanelli MN. Chiaramonte N, et al. Among authors: braconi l. J Enzyme Inhib Med Chem. 2020 Dec;35(1):1003-1010. doi: 10.1080/14756366.2020.1749602. J Enzyme Inhib Med Chem. 2020. PMID: 32336172 Free PMC article.

8

1-benzyl-1,4-diazepane reduces the efflux of resistance-nodulation-cell division pumps in Escherichia coli.

Casalone E, Vignolini T, Braconi L, Gardini L, Capitanio M, Pavone FS, Dei S, Teodori E. Casalone E, et al. Among authors: braconi l. Future Microbiol. 2020 Jul;15:987-999. doi: 10.2217/fmb-2019-0296. Epub 2020 Aug 25. Future Microbiol. 2020. PMID: 32840130

9

Characterization of substituted piperazines able to reverse MDR in Escherichia coli strains overexpressing resistance-nodulation-cell division (RND) efflux pumps.

Casalone E, Vignolini T, Braconi L, Gardini L, Capitanio M, Pavone FS, Giovannelli L, Dei S, Teodori E. Casalone E, et al. Among authors: braconi l. J Antimicrob Chemother. 2022 Feb 2;77(2):413-424. doi: 10.1093/jac/dkab388. J Antimicrob Chemother. 2022. PMID: 34747445

10

2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity.

Chiaramonte N, Angeli A, Sgambellone S, Bonardi A, Nocentini A, Bartolucci G, Braconi L, Dei S, Lucarini L, Teodori E, Gratteri P, Wünsch B, Supuran CT, Romanelli MN. Chiaramonte N, et al. Among authors: braconi l. Eur J Med Chem. 2022 Jan 15;228:114026. doi: 10.1016/j.ejmech.2021.114026. Epub 2021 Dec 4. Eur J Med Chem. 2022. PMID: 34920169

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