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Eugenol derivatives with 1,2,3-triazole moieties: Oral treatment of cutaneous leishmaniasis and a quantitative structure-activity relationship model for their leishmanicidal activity.
Exp Parasitol. 2022 Jul;238:108269. doi: 10.1016/j.exppara.2022.108269. Epub 2022 May 5.
Exp Parasitol. 2022.
PMID: 35526574
Chalcones identify cTXNPx as a potential antileishmanial drug target.
Escrivani DO, Charlton RL, Caruso MB, Burle-Caldas GA, Borsodi MPG, Zingali RB, Arruda-Costa N, Palmeira-Mello MV, de Jesus JB, Souza AMT, Abrahim-Vieira B, Freitag-Pohl S, Pohl E, Denny PW, Rossi-Bergmann B, Steel PG.
Escrivani DO, et al. Among authors: borsodi mpg.
PLoS Negl Trop Dis. 2021 Nov 15;15(11):e0009951. doi: 10.1371/journal.pntd.0009951. eCollection 2021 Nov.
PLoS Negl Trop Dis. 2021.
PMID: 34780470
Free PMC article.
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Leishmanicidal and cytotoxic activities and 4D-QSAR of 2-arylidene indan-1,3-diones.
de Souza APM, Costa MCA, de Aguiar AR, Bressan GC, de Almeida Lima GD, Lima WP, Borsodi MPG, Bergmann BR, Ferreira MMC, Teixeira RR.
de Souza APM, et al. Among authors: borsodi mpg.
Arch Pharm (Weinheim). 2021 Oct;354(10):e2100081. doi: 10.1002/ardp.202100081. Epub 2021 Jul 29.
Arch Pharm (Weinheim). 2021.
PMID: 34323311
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Antileishmanial Chemotherapy through Clemastine Fumarate Mediated Inhibition of the Leishmania Inositol Phosphorylceramide Synthase.
Mina JGM, Charlton RL, Alpizar-Sosa E, Escrivani DO, Brown C, Alqaisi A, Borsodi MPG, Figueiredo CP, de Lima EV, Dickie EA, Wei W, Coutinho-Silva R, Merritt A, Smith TK, Barrett MP, Rossi-Bergmann B, Denny PW, Steel PG.
Mina JGM, et al. Among authors: borsodi mpg.
ACS Infect Dis. 2021 Jan 8;7(1):47-63. doi: 10.1021/acsinfecdis.0c00546. Epub 2020 Dec 8.
ACS Infect Dis. 2021.
PMID: 33291887
Free PMC article.
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Nanoparticles Loaded with a New Thiourea Derivative: Development and In vitro Evaluation Against Leishmania amazonensis.
Meireles PW, de Souza DPB, Rezende MG, Borsodi MPG, de Oliveira DE, da Silva LCRP, de Souza AMT, Viana GM, Rodrigues CR, do Carmo FA, de Sousa VP, Rossi-Bergmann B, Cabral LM.
Meireles PW, et al. Among authors: borsodi mpg.
Curr Drug Deliv. 2020;17(8):694-702. doi: 10.2174/1567201817666200704132348.
Curr Drug Deliv. 2020.
PMID: 32621717
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Leishmanicidal activity of Piper marginatum Jacq. from Santarém-PA against Leishmania amazonensis.
Macêdo CG, Fonseca MYN, Caldeira AD, Castro SP, Pacienza-Lima W, Borsodi MPG, Sartoratto A, da Silva MN, Salgado CG, Rossi-Bergmann B, Castro KCF.
Macêdo CG, et al. Among authors: borsodi mpg.
Exp Parasitol. 2020 Mar;210:107847. doi: 10.1016/j.exppara.2020.107847. Epub 2020 Jan 28.
Exp Parasitol. 2020.
PMID: 32004535
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Synthesis and leishmanicidal activity of eugenol derivatives bearing 1,2,3-triazole functionalities.
Teixeira RR, Gazolla PAR, da Silva AM, Borsodi MPG, Bergmann BR, Ferreira RS, Vaz BG, Vasconcelos GA, Lima WP.
Teixeira RR, et al. Among authors: borsodi mpg.
Eur J Med Chem. 2018 Feb 25;146:274-286. doi: 10.1016/j.ejmech.2018.01.046. Epub 2018 Feb 4.
Eur J Med Chem. 2018.
PMID: 29407957
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Optimization of Aqueous Extraction from Kalanchoe pinnata Leaves to Obtain the Highest Content of an Anti-inflammatory Flavonoid using a Response Surface Model.
Dos Santos Nascimento LB, de Aguiar PF, Leal-Costa MV, Coutinho MAS, Borsodi MPG, Rossi-Bergmann B, Tavares ES, Costa SS.
Dos Santos Nascimento LB, et al. Among authors: borsodi mpg.
Phytochem Anal. 2018 May;29(3):308-315. doi: 10.1002/pca.2744. Epub 2018 Jan 19.
Phytochem Anal. 2018.
PMID: 29349835
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