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Discovery of a septin-4 covalent binder with antimetastatic activity in a mouse model of melanoma.
Bioorg Chem. 2024 Mar;144:107164. doi: 10.1016/j.bioorg.2024.107164. Epub 2024 Jan 29.
Bioorg Chem. 2024.
PMID: 38306824
Free article.
Discovery of a novel 1,3,4-oxadiazol-2-one-based NLRP3 inhibitor as a pharmacological agent to mitigate cardiac and metabolic complications in an experimental model of diet-induced metaflammation.
Gastaldi S, Rocca C, Gianquinto E, Granieri MC, Boscaro V, Blua F, Rolando B, Marini E, Gallicchio M, De Bartolo A, Romeo N, Mazza R, Fedele F, Pagliaro P, Penna C, Spyrakis F, Bertinaria M, Angelone T.
Gastaldi S, et al. Among authors: blua f.
Eur J Med Chem. 2023 Sep 5;257:115542. doi: 10.1016/j.ejmech.2023.115542. Epub 2023 Jun 2.
Eur J Med Chem. 2023.
PMID: 37290185
Free article.
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Comparative Study of Different H2S Donors as Vasodilators and Attenuators of Superoxide-Induced Endothelial Damage.
Marini E, Rolando B, Sodano F, Blua F, Concina G, Guglielmo S, Lazzarato L, Chegaev K.
Marini E, et al. Among authors: blua f.
Antioxidants (Basel). 2023 Feb 1;12(2):344. doi: 10.3390/antiox12020344.
Antioxidants (Basel). 2023.
PMID: 36829903
Free PMC article.
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Investigation into the Use of Encorafenib to Develop Potential PROTACs Directed against BRAFV600E Protein.
Marini E, Marino M, Gionfriddo G, Maione F, Pandini M, Oddo D, Giorgis M, Rolando B, Blua F, Gastaldi S, Marchiò S, Kovachka S, Spyrakis F, Gianquinto E, Di Nicolantonio F, Bertinaria M.
Marini E, et al. Among authors: blua f.
Molecules. 2022 Dec 3;27(23):8513. doi: 10.3390/molecules27238513.
Molecules. 2022.
PMID: 36500607
Free PMC article.
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Chemical Modulation of the 1-(Piperidin-4-yl)-1,3-dihydro-2H-benzo[d]imidazole-2-one Scaffold as a Novel NLRP3 Inhibitor.
Gastaldi S, Boscaro V, Gianquinto E, Sandall CF, Giorgis M, Marini E, Blua F, Gallicchio M, Spyrakis F, MacDonald JA, Bertinaria M.
Gastaldi S, et al. Among authors: blua f.
Molecules. 2021 Jun 29;26(13):3975. doi: 10.3390/molecules26133975.
Molecules. 2021.
PMID: 34209843
Free PMC article.
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