Bjørn-Yoshimoto WE - Search Results

1

Ligand selectivity hotspots in serotonin GPCRs.

Simon IA, Bjørn-Yoshimoto WE, Harpsøe K, Iliadis S, Svensson B, Jensen AA, Gloriam DE. Simon IA, et al. Among authors: bjorn yoshimoto we. Trends Pharmacol Sci. 2023 Dec;44(12):978-990. doi: 10.1016/j.tips.2023.09.012. Epub 2023 Oct 31. Trends Pharmacol Sci. 2023. PMID: 37914598 Free article. Review.

2

5-HT_2C Receptor Structures Reveal the Structural Basis of GPCR Polypharmacology.

Peng Y, McCorvy JD, Harpsøe K, Lansu K, Yuan S, Popov P, Qu L, Pu M, Che T, Nikolajsen LF, Huang XP, Wu Y, Shen L, Bjørn-Yoshimoto WE, Ding K, Wacker D, Han GW, Cheng J, Katritch V, Jensen AA, Hanson MA, Zhao S, Gloriam DE, Roth BL, Stevens RC, Liu ZJ. Peng Y, et al. Among authors: bjorn yoshimoto we. Cell. 2018 Feb 8;172(4):719-730.e14. doi: 10.1016/j.cell.2018.01.001. Epub 2018 Feb 1. Cell. 2018. PMID: 29398112 Free PMC article.

3

Excitatory amino acid transporters: recent insights into molecular mechanisms, novel modes of modulation and new therapeutic possibilities.

Jensen AA, Fahlke C, Bjørn-Yoshimoto WE, Bunch L. Jensen AA, et al. Curr Opin Pharmacol. 2015 Feb;20:116-23. doi: 10.1016/j.coph.2014.10.008. Epub 2014 Nov 5. Curr Opin Pharmacol. 2015. PMID: 25466154 Review.

4

β-Sulfonamido Functionalized Aspartate Analogues as Excitatory Amino Acid Transporter Inhibitors: Distinct Subtype Selectivity Profiles Arising from Subtle Structural Differences.

Hansen JC, Bjørn-Yoshimoto WE, Bisballe N, Nielsen B, Jensen AA, Bunch L. Hansen JC, et al. J Med Chem. 2016 Oct 13;59(19):8771-8786. doi: 10.1021/acs.jmedchem.6b01066. Epub 2016 Sep 16. J Med Chem. 2016. PMID: 27636002

5

Identification and Structure-Activity Relationship Study of Imidazo[1,2-a]pyridine-3-amines as First Selective Inhibitors of Excitatory Amino Acid Transporter Subtype 3 (EAAT3).

Wu P, Bjørn-Yoshimoto WE, Staudt M, Jensen AA, Bunch L. Wu P, et al. Among authors: bjorn yoshimoto we. ACS Chem Neurosci. 2019 Oct 16;10(10):4414-4429. doi: 10.1021/acschemneuro.9b00447. Epub 2019 Oct 1. ACS Chem Neurosci. 2019. PMID: 31573179

6

Identification of a New Class of Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors Followed by a Structure-Activity Relationship Study.

Hansen SW, Erichsen MN, Fu B, Bjørn-Yoshimoto WE, Abrahamsen B, Hansen JC, Jensen AA, Bunch L. Hansen SW, et al. J Med Chem. 2016 Oct 13;59(19):8757-8770. doi: 10.1021/acs.jmedchem.6b01058. Epub 2016 Sep 14. J Med Chem. 2016. PMID: 27626828

7

New Insight into the Structure-Activity Relationships of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors UCPH-101 and UCPH-102.

Hansen SW, Erichsen MN, Huynh TH, Ruiz JA, Haym I, Bjørn-Yoshimoto WE, Abrahamsen B, Hansen J, Storgaard M, Eriksen AL, Jensen AA, Bunch L. Hansen SW, et al. ChemMedChem. 2016 Feb 17;11(4):382-402. doi: 10.1002/cmdc.201500525. Epub 2016 Jan 12. ChemMedChem. 2016. PMID: 26757239

8

Bioavailability Studies and in vitro Profiling of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitor UCPH-102.

Haym I, Huynh TH, Hansen SW, Pedersen MH, Ruiz JA, Erichsen MN, Gynther M, Bjørn-Yoshimoto WE, Abrahamsen B, Bastlund JF, Bundgaard C, Eriksen AL, Jensen AA, Bunch L. Haym I, et al. ChemMedChem. 2016 Feb 17;11(4):403-19. doi: 10.1002/cmdc.201500527. Epub 2016 Jan 21. ChemMedChem. 2016. PMID: 26797816 Free article.

9

Design and Synthesis of 2,3- trans-Proline Analogues as Ligands for Ionotropic Glutamate Receptors and Excitatory Amino Acid Transporters.

Poulie CBM, Alcaide A, Krell-Jørgensen M, Larsen Y, Astier E, Bjørn-Yoshimoto WE, Yi F, Syrenne JT, Storgaard M, Nielsen B, Frydenvang KA, Jensen AA, Hansen KB, Pickering DS, Bunch L. Poulie CBM, et al. Among authors: bjorn yoshimoto we. ACS Chem Neurosci. 2019 Jun 19;10(6):2989-3007. doi: 10.1021/acschemneuro.9b00205. Epub 2019 May 24. ACS Chem Neurosci. 2019. PMID: 31124660 Free PMC article.

10

(S)-2-Mercaptohistidine: A First Selective Orthosteric GluK3 Antagonist.

Poulie CBM, Larsen Y, Leteneur C, Barthet G, Bjørn-Yoshimoto WE, Malhaire F, Nielsen B, Pin JP, Mulle C, Pickering DS, Bunch L. Poulie CBM, et al. Among authors: bjorn yoshimoto we. ACS Chem Neurosci. 2022 May 18;13(10):1580-1587. doi: 10.1021/acschemneuro.2c00162. Epub 2022 Apr 27. ACS Chem Neurosci. 2022. PMID: 35475632

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