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An ultra-high-affinity small organic ligand of fibroblast activation protein for tumor-targeting applications.
Proc Natl Acad Sci U S A. 2021 Apr 20;118(16):e2101852118. doi: 10.1073/pnas.2101852118.
Proc Natl Acad Sci U S A. 2021.
PMID: 33850024
Free PMC article.
Deep Learning Approach for the Discovery of Tumor-Targeting Small Organic Ligands from DNA-Encoded Chemical Libraries.
Torng W, Biancofiore I, Oehler S, Xu J, Xu J, Watson I, Masina B, Prati L, Favalli N, Bassi G, Neri D, Cazzamalli S, Feng JA.
Torng W, et al. Among authors: biancofiore i.
ACS Omega. 2023 Jul 6;8(28):25090-25100. doi: 10.1021/acsomega.3c01775. eCollection 2023 Jul 18.
ACS Omega. 2023.
PMID: 37483198
Free PMC article.
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Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 Interaction.
Ontoria JM, Biancofiore I, Fezzardi P, Ferrigno F, Torrente E, Colarusso S, Bianchi E, Andreini M, Patsilinakos A, Kempf G, Augustin M, Steinbacher S, Summa V, Pacifici R, Muñoz-Sanjuan I, Park L, Bresciani A, Dominguez C, Sherman LT, Harper S.
Ontoria JM, et al. Among authors: biancofiore i.
ACS Med Chem Lett. 2020 Apr 3;11(5):740-746. doi: 10.1021/acsmedchemlett.9b00594. eCollection 2020 May 14.
ACS Med Chem Lett. 2020.
PMID: 32435379
Free PMC article.
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Optimization of 2-(1H-imidazo-2-yl)piperazines series of Trypanosoma brucei growth inhibitors as potential treatment for the second stage of HAT.
Ciammaichella A, Ferrigno F, Basta A, D'Amico M, Biancofiore I, Nardi V, Ponzi S, Graziani R, Gennari N, Vittoria Orsale M, Fini I, Paonessa G, Summa V, Harper S, Ontoria JM.
Ciammaichella A, et al. Among authors: biancofiore i.
Bioorg Med Chem Lett. 2020 Jun 15;30(12):127207. doi: 10.1016/j.bmcl.2020.127207. Epub 2020 Apr 21.
Bioorg Med Chem Lett. 2020.
PMID: 32354566
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Sulphide as a leaving group: highly stereoselective bromination of alkyl phenyl sulphides.
Canestrari D, Cioffi C, Biancofiore I, Lancianesi S, Ghisu L, Ruether M, O'Brien J, Adamo MFA, Ibrahim H.
Canestrari D, et al. Among authors: biancofiore i.
Chem Sci. 2019 Aug 16;10(39):9042-9050. doi: 10.1039/c9sc03560e. eCollection 2019 Oct 21.
Chem Sci. 2019.
PMID: 31827746
Free PMC article.
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Improved Selective Class I HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and Benzamides.
Bresciani A, Ontoria JM, Biancofiore I, Cellucci A, Ciammaichella A, Di Marco A, Ferrigno F, Francone A, Malancona S, Monteagudo E, Nizi E, Pace P, Ponzi S, Rossetti I, Veneziano M, Summa V, Harper S.
Bresciani A, et al. Among authors: biancofiore i.
ACS Med Chem Lett. 2018 Nov 27;10(4):481-486. doi: 10.1021/acsmedchemlett.8b00517. eCollection 2019 Apr 11.
ACS Med Chem Lett. 2018.
PMID: 30996783
Free PMC article.
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Discovery of 2-(1H-imidazo-2-yl)piperazines as a new class of potent and non-cytotoxic inhibitors of Trypanosoma brucei growth in vitro.
Ferrigno F, Biancofiore I, Malancona S, Ponzi S, Paonessa G, Graziani R, Bresciani A, Gennari N, Di Marco A, Kaiser M, Summa V, Harper S, Ontoria JM.
Ferrigno F, et al. Among authors: biancofiore i.
Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3689-3692. doi: 10.1016/j.bmcl.2018.10.028. Epub 2018 Oct 22.
Bioorg Med Chem Lett. 2018.
PMID: 30482621
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Discovery of a Selective Series of Inhibitors of Plasmodium falciparum HDACs.
Ontoria JM, Paonessa G, Ponzi S, Ferrigno F, Nizi E, Biancofiore I, Malancona S, Graziani R, Roberts D, Willis P, Bresciani A, Gennari N, Cecchetti O, Monteagudo E, Orsale MV, Veneziano M, Di Marco A, Cellucci A, Laufer R, Altamura S, Summa V, Harper S.
Ontoria JM, et al. Among authors: biancofiore i.
ACS Med Chem Lett. 2016 Mar 5;7(5):454-9. doi: 10.1021/acsmedchemlett.5b00468. eCollection 2016 May 12.
ACS Med Chem Lett. 2016.
PMID: 27190592
Free PMC article.
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