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Native metabotropic glutamate receptor 4 depresses synaptic transmission through an unusual Gαq transduction pathway.
Neuropharmacology. 2017 Jul 15;121:247-260. doi: 10.1016/j.neuropharm.2017.04.036. Epub 2017 Apr 26.
Neuropharmacology. 2017.
PMID: 28456688
A new signalling pathway for parallel fibre presynaptic type 4 metabotropic glutamate receptors (mGluR4) in the rat cerebellar cortex.
Abitbol K, McLean H, Bessiron T, Daniel H.
Abitbol K, et al. Among authors: bessiron t.
J Physiol. 2012 Jul 1;590(13):2977-94. doi: 10.1113/jphysiol.2012.232074. Epub 2012 May 8.
J Physiol. 2012.
PMID: 22570379
Free PMC article.
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A novel selective metabotropic glutamate receptor 4 agonist reveals new possibilities for developing subtype selective ligands with therapeutic potential.
Goudet C, Vilar B, Courtiol T, Deltheil T, Bessiron T, Brabet I, Oueslati N, Rigault D, Bertrand HO, McLean H, Daniel H, Amalric M, Acher F, Pin JP.
Goudet C, et al. Among authors: bessiron t.
FASEB J. 2012 Apr;26(4):1682-93. doi: 10.1096/fj.11-195941. Epub 2012 Jan 5.
FASEB J. 2012.
PMID: 22223752
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Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites.
Selvam C, Lemasson IA, Brabet I, Oueslati N, Karaman B, Cabaye A, Tora AS, Commare B, Courtiol T, Cesarini S, McCort-Tranchepain I, Rigault D, Mony L, Bessiron T, McLean H, Leroux FR, Colobert F, Daniel H, Goupil-Lamy A, Bertrand HO, Goudet C, Pin JP, Acher FC.
Selvam C, et al. Among authors: bessiron t.
J Med Chem. 2018 Mar 8;61(5):1969-1989. doi: 10.1021/acs.jmedchem.7b01438. Epub 2018 Feb 14.
J Med Chem. 2018.
PMID: 29397723
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