Berthelot P - Search Results

1

New Quinoxaline Derivatives as Dual Pim-1/2 Kinase Inhibitors: Design, Synthesis and Biological Evaluation.

Oyallon B, Brachet-Botineau M, Logé C, Robert T, Bach S, Ibrahim S, Raoul W, Croix C, Berthelot P, Guillon J, Pinaud N, Gouilleux F, Viaud-Massuard MC, Denevault-Sabourin C. Oyallon B, et al. Among authors: berthelot p. Molecules. 2021 Feb 6;26(4):867. doi: 10.3390/molecules26040867. Molecules. 2021. PMID: 33562106 Free PMC article.

2

Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors.

Oyallon B, Brachet-Botineau M, Logé C, Bonnet P, Souab M, Robert T, Ruchaud S, Bach S, Berthelot P, Gouilleux F, Viaud-Massuard MC, Denevault-Sabourin C. Oyallon B, et al. Among authors: berthelot p. Eur J Med Chem. 2018 Jun 25;154:101-109. doi: 10.1016/j.ejmech.2018.04.056. Epub 2018 May 11. Eur J Med Chem. 2018. PMID: 29778892

3

Docking study of ligands into the colchicine binding site of tubulin.

Farce A, Loge C, Gallet S, Lebegue N, Carato P, Chavatte P, Berthelot P, Lesieur D. Farce A, et al. Among authors: berthelot p. J Enzyme Inhib Med Chem. 2004 Dec;19(6):541-7. doi: 10.1080/14756360412331280545. J Enzyme Inhib Med Chem. 2004. PMID: 15662957

4

Synthesis, biological evaluation and docking studies of 4-amino-tetrahydroquinazolino[3,2-e]purine derivatives.

Verones V, Flouquet N, Farce A, Carato P, Leonce S, Pfeiffer B, Berthelot P, Lebegue N. Verones V, et al. Among authors: berthelot p. Eur J Med Chem. 2010 Dec;45(12):5678-84. doi: 10.1016/j.ejmech.2010.09.022. Epub 2010 Sep 17. Eur J Med Chem. 2010. PMID: 20884092

5

Novel conformationally constrained analogues of agomelatine as new melatoninergic ligands.

Rami M, Landagaray E, Ettaoussi M, Boukhalfa K, Caignard DH, Delagrange P, Berthelot P, Yous S. Rami M, et al. Among authors: berthelot p. Molecules. 2012 Dec 24;18(1):154-66. doi: 10.3390/molecules18010154. Molecules. 2012. PMID: 23262445 Free PMC article.

6

Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3.

Leclerc V, Ettaoussi M, Rami M, Farce A, Boutin JA, Delagrange P, Caignard DH, Renard P, Berthelot P, Yous S. Leclerc V, et al. Among authors: berthelot p. Eur J Med Chem. 2011 May;46(5):1622-9. doi: 10.1016/j.ejmech.2011.02.010. Epub 2011 Feb 15. Eur J Med Chem. 2011. PMID: 21377769

7

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands.

Mésangeau C, Pérès B, Descamps-François C, Chavatte P, Audinot V, Coumailleau S, Boutin JA, Delagrange P, Bennejean C, Renard P, Caignard DH, Berthelot P, Yous S. Mésangeau C, et al. Among authors: berthelot p. Bioorg Med Chem. 2010 May 15;18(10):3426-36. doi: 10.1016/j.bmc.2010.04.008. Epub 2010 Apr 7. Bioorg Med Chem. 2010. PMID: 20444610

8

Design, synthesis and pharmacological evaluation of new series of naphthalenic analogues as melatoninergic (MT1/MT2) and serotoninergic 5-HT2C dual ligands (I).

Ettaoussi M, Sabaouni A, Rami M, Boutin JA, Delagrange P, Renard P, Spedding M, Caignard DH, Berthelot P, Yous S. Ettaoussi M, et al. Among authors: berthelot p. Eur J Med Chem. 2012 Mar;49:310-23. doi: 10.1016/j.ejmech.2012.01.027. Epub 2012 Jan 20. Eur J Med Chem. 2012. PMID: 22301214

9

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Part II.

Durieux S, Chanu A, Bochu C, Audinot V, Coumailleau S, Boutin JA, Delagrange P, Caignard DH, Bennejean C, Renard P, Lesieur D, Berthelot P, Yous S. Durieux S, et al. Among authors: berthelot p. Bioorg Med Chem. 2009 Apr 15;17(8):2963-74. doi: 10.1016/j.bmc.2009.03.023. Epub 2009 Mar 18. Bioorg Med Chem. 2009. PMID: 19329323

10

New antiproliferative benzoindolinothiazepines derivatives.

Laconde G, Depreux P, Berthelot P, Pommery N, Hénichart JP. Laconde G, et al. Among authors: berthelot p. Eur J Med Chem. 2005 Feb;40(2):167-72. doi: 10.1016/j.ejmech.2004.10.008. Eur J Med Chem. 2005. PMID: 15694651

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